| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA650823 | B | Inhibition of [3H]-Ro- 15-1788 binding to GABA-A benzodiazepine receptor of bovine brain membranes | Bos taurus | 22 | cell membrane format | Scientific Literature | ||
| 2. | ALA652658 | B | Inhibition of [3H]- flumazenil binding to benzodiazepine receptor in bovine brain membranes | 40 | cell membrane format | Scientific Literature | |||
| 3. | ALA652660 | B | Ratio of Ki with out GABA and with GABA | 31 | protein complex format | Scientific Literature | |||
| 4. | ALA681818 | B | Inhibition of TBPS binding to GABA-A receptor of bovine brain membranes at 0.5 uM relative to clonazepam | Bos taurus | 10 | cell membrane format | Scientific Literature | ||
| 5. | ALA720987 | F | Antagonistic effect against PTZ (80 mg/kg, sc) convulsant action in mice | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 6. | ALA727835 | F | Antagonistic effect against the anticonvulsant Diazepam (2.5 mg/kg, ip) effect in mice after PTZ (80mg/kg, sc) dose, ineffective to 250 mg/kg | Mus musculus | 4 | organism-based format | Scientific Literature | ||
| 7. | ALA727676 | F | Convulsant effect in mice following subconvulsant PTZ(40 mg/kg, sc) dose, ineffective to 250 mg/kg | Mus musculus | 5 | organism-based format | Scientific Literature | ||
| 8. | ALA822945 | B | Inhibition of [3H]flumazenil binding to rat alpha-1-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cells | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA823760 | B | Inhibition of [3H]flumazenil binding to rat alpha-3-beta-2-gamma-2 GABA-A receptor subunits expressed in HEK293 cells | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA818518 | B | Inhibition of [3H]flumazenil binding to rat alpha-5-beta-3-gamma-2 GABA-A receptor subunits expressed in HEK293 cells | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA841636 | B | Relative binding to GABA-A receptor in the presence and absence of GABA (GABA shift), Ki(-GABA)/Ki(+GABA) | Bos taurus | 13 | protein complex format | Scientific Literature | ||
| 12. | ALA848601 | B | Ratio of Ki with out GABA and with GABA | 8 | protein complex format | Scientific Literature |
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