# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA650182 | B | Percent inhibition of [3H]- Diazepam binding to GABA-A Benzodiazepine receptor of rat frontal cortex membranes (ND = no data) | Rattus norvegicus | 7 | ALA1122999 | cell membrane format | Scientific Literature | |
2. | ALA657004 | F | BMC-sensitive inhibitory effect on cat spinal neurons relative to that of GABA was expressed in vivo as relative potency; Greater activity | Felis catus | 3 | ALA1122838 | organism-based format | Scientific Literature | |
3. | ALA681334 | B | Displacement of [3H]gamma-amino butyric acid from Gamma-aminobutyric acid (GABA-A) receptor of human cerebellar cortex preparation | Homo sapiens | 6 | ALA1121465 | assay format | Scientific Literature | |
4. | ALA682053 | B | Percent displacement of [3H]GABA at Gamma-aminobutyric acid receptor of rat brain membranes at 0.01 uM | Rattus norvegicus | 2 | ALA1121865 | cell membrane format | Scientific Literature | |
5. | ALA679668 | F | Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytes | Homo sapiens | 1 | ALA1133003 | cell-based format | Scientific Literature | |
6. | ALA679669 | F | Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytes | Homo sapiens | 1 | ALA1133003 | cell-based format | Scientific Literature | |
7. | ALA681130 | B | Displacement of [3H]gamma-aminobutyric acid from sodium-independent Gamma-aminobutyric acid (GABA-A) receptor synaptic membrane binding sites from rat brain tissue | Rattus norvegicus | 3 | ALA1121547 | assay format | Scientific Literature | |
8. | ALA681136 | B | In vitro inhibition of [3H]GABA binding to Gamma-aminobutyric acid receptor of rat brain synaptic membranes | Rattus norvegicus | 5 | ALA1122838 | cell membrane format | Scientific Literature | |
9. | ALA681137 | B | In vitro inhibition of [3H]P4S binding to Gamma-aminobutyric acid receptor of rat brain synaptic membranes | Rattus norvegicus | 7 | ALA1122838 | cell membrane format | Scientific Literature | |
10. | ALA681138 | B | In vitro inhibition of [3H]THIP binding to Gamma-aminobutyric acid receptor in rat brain synaptic membranes | Rattus norvegicus | 7 | ALA1122838 | cell membrane format | Scientific Literature | |
11. | ALA681302 | B | Displacement of [3H]- muscimol in cerebral tissue of male rats | Rattus norvegicus | 3 | ALA1122920 | protein complex format | Scientific Literature | |
12. | ALA681304 | B | Displacement of [3H]- muscimol from GABA-A receptor from rat cerebellum membrane at 0.003-0.006 uM | Rattus norvegicus | 1 | ALA1122999 | tissue-based format | Scientific Literature | |
13. | ALA680229 | B | Displacement of [3H]gamma-amino butyric acid from Gamma-aminobutyric acid (GABA-A) receptor of rat ganglion neurons | Rattus norvegicus | 6 | ALA1121465 | protein complex format | Scientific Literature | |
14. | ALA681817 | B | Relative binding affinity for sodium-independent Gamma-aminobutyric acid receptor synaptic membrane binding site in rat brain tissue | Rattus norvegicus | 4 | ALA1121547 | tissue-based format | Scientific Literature | |
15. | ALA681240 | B | Displacement of [3H]GABA from Gamma-aminobutyric acid A receptor ofrat brain membranes | Rattus norvegicus | 12 | ALA1123925 | assay format | Scientific Literature | |
16. | ALA681241 | B | Inhibition against Gamma-aminobutyric acid A (GABA-A) receptor | Rattus norvegicus | 3 | ALA1133561 | protein complex format | Scientific Literature | |
17. | ALA681949 | F | Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations. | Bos taurus | 12 | ALA1125342 | tissue-based format | Scientific Literature | |
18. | ALA681951 | B | Binding affinity in vivo for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]-GABA agonist from rat brain preparations after iv injection. | Bos taurus | 23 | ALA1125342 | organism-based format | Scientific Literature | |
19. | ALA679565 | B | Affinity for GGABA-A receptor alpha by inhibiting binding of [3H]muscimol to rat brain synaptosomes | 2 | ALA1135459 | subcellular format | Scientific Literature | ||
20. | ALA677637 | B | Percent of enzyme inhibition by Gamma-amino-N-butyrate transaminase assay method ND means no data | 1 | ALA1122999 | single protein format | Scientific Literature |