| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA679557 | B | Inhibitory activity against human sodium and chloride dependent GABA transporter 3 | 25 | ALA1127589 | single protein format | Scientific Literature | ||
| 2. | ALA806333 | B | Inhibitory activity against human GABA transporter-1 (hGAT1) | 28 | ALA1127589 | single protein format | Scientific Literature | ||
| 3. | ALA806336 | B | Compound was evaluated for inhibitory activity against human GABA transporter (hBGT-1)at 100 uM concentration | 5 | ALA1127589 | single protein format | Scientific Literature | ||
| 4. | ALA809055 | B | Inhibitory activity against rat GABA transporter-2 (rGAT2) | 25 | ALA1127589 | single protein format | Scientific Literature | ||
| 5. | ALA1776005 | B | Inhibition of human GAT1-mediated GABA uptake | Homo sapiens | 1 | ALA1773002 | single protein format | Scientific Literature | |
| 6. | ALA1776006 | B | Inhibition of human BGT1-mediated GABA uptake at 100 uM | Homo sapiens | 1 | ALA1773002 | single protein format | Scientific Literature | |
| 7. | ALA1776007 | B | Inhibition of rat GAT2-mediated GABA uptake | Rattus norvegicus | 1 | ALA1773002 | single protein format | Scientific Literature | |
| 8. | ALA1776008 | B | Inhibition of human GAT3-mediated GABA uptake | Homo sapiens | 1 | ALA1773002 | single protein format | Scientific Literature | |
| 9. | ALA3877711 | B | Inhibition of mouse GAT3 expressed in HEK293 cells assessed as decrease in [3H]GABA uptake preincubated for 25 mins followed by [3H]GABA addition measured after 4 mins by liquid scintillation counter method | Mus musculus | 14 | ALA3877251 | cell-based format | Scientific Literature | |
| 10. | ALA3877712 | B | Inhibition of mouse GAT4 expressed in HEK293 cells assessed as decrease in [3H]GABA uptake preincubated for 25 mins followed by [3H]GABA addition measured after 4 mins by liquid scintillation counter method | Mus musculus | 13 | ALA3877251 | cell-based format | Scientific Literature | |
| 11. | ALA3877713 | B | Inhibition of human GAT-1 expressed in thymidine kinase deficient mouse LM cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation counter method | Homo sapiens | 1 | ALA3877251 | cell-based format | Scientific Literature | |
| 12. | ALA3877714 | B | Inhibition of human BGT-1 expressed in thymidine kinase deficient mouse LM cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation counter method | Homo sapiens | 1 | ALA3877251 | cell-based format | Scientific Literature | |
| 13. | ALA3877715 | B | Inhibition of rat GAT-2 expressed in thymidine kinase deficient mouse LM cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation counter method | Rattus norvegicus | 1 | ALA3877251 | cell-based format | Scientific Literature | |
| 14. | ALA3877716 | B | Inhibition of human GAT-3 expressed in thymidine kinase deficient mouse LM cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation counter method | Homo sapiens | 1 | ALA3877251 | cell-based format | Scientific Literature | |
| 15. | ALA3877720 | B | Inhibition of mouse GAT1 expressed in HEK293 cells assessed as decrease in [3H]GABA uptake at 100 uM preincubated for 25 mins followed by [3H]GABA addition measured after 4 mins by liquid scintillation counter method | Mus musculus | 15 | ALA3877251 | cell-based format | Scientific Literature | |
| 16. | ALA3877721 | B | Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptake at 100 uM preincubated for 25 mins followed by [3H]GABA addition measured after 10 mins by liquid scintillation counter method | Mus musculus | 12 | ALA3877251 | cell-based format | Scientific Literature |
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