# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3539957 | ADME | Inhibition of recombinant human C-terminal His-tagged UGT1A10 after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
2. | ALA3539958 | ADME | Inhibition of recombinant human C-terminal His-tagged UGT2B7 after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
3. | ALA3537416 | ADME | Drug metabolism in human liver microsomes assessed as 16-epiestriol-3-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | assay format | Scientific Literature | |
4. | ALA3537417 | ADME | Drug metabolism in human liver microsomes assessed as 16-epiestriol-16-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | assay format | Scientific Literature | |
5. | ALA3537756 | ADME | Drug metabolism in human intestine microsomes assessed as 16-epiestriol-3-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | assay format | Scientific Literature | |
6. | ALA3537757 | ADME | Drug metabolism in human intestine microsomes assessed as 16-epiestriol-16-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | assay format | Scientific Literature | |
7. | ALA3537758 | ADME | Drug metabolism in human intestine microsomes assessed as 16-epiestriol-17-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | assay format | Scientific Literature | |
8. | ALA3532613 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT2B7-mediated 16-epiestriol-16-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
9. | ALA3532616 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT2B7-mediated 16-epiestriol-16-glucuronide formation at 5 mg after 5 hrs by NMR spectroscopic analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
10. | ALA3532618 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT2B17-mediated 16-epiestriol-17-glucuronide formation at 5 mg after 5 hrs by NMR spectroscopic analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
11. | ALA3532969 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT1A10-mediated 16-epiestriol-3-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
12. | ALA3532970 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT1A1-mediated 16-epiestriol-3-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
13. | ALA3532971 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT1A7-mediated 16-epiestriol-3-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
14. | ALA3532972 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT1A8-mediated 16-epiestriol-3-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
15. | ALA3532973 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT2B15-mediated 16-epiestriol-3-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
16. | ALA3532974 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT1A3-mediated 16-epiestriol-16-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
17. | ALA3532975 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT2A1-mediated 16-epiestriol-16-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
18. | ALA3532976 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT2B4-mediated 16-epiestriol-16-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
19. | ALA3532977 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT2B17-mediated 16-epiestriol-16-glucuronide formation after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature | |
20. | ALA3532978 | ADME | Drug metabolism assessed as recombinant human C-terminal His-tagged UGT1A4-mediated 16-epiestriol-16-glucuronide formation at 200 uM after 15 to 60 mins by HPLC analysis in presence of UDPGA | Homo sapiens | 1 | ALA3525985 | single protein format | Scientific Literature |