| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1919073 | B | Inhibition of human placental microsomal 17beta-HSD2 at 1 uM by HPLC analysis | Homo sapiens | 21 | assay format | Scientific Literature | ||
| 2. | ALA1919074 | B | Inhibition of human placental cytosolic 17beta-HSD1 at 1 uM by HPLC analysis | Homo sapiens | 21 | assay format | Scientific Literature | ||
| 3. | ALA1919075 | B | Inhibition of human placental microsomal 17beta-HSD2 using [3H]E2 as substrate by HPLC analysis | Homo sapiens | 9 | assay format | Scientific Literature | ||
| 4. | ALA1919076 | B | Inhibition of human placental cytosolic 17beta-HSD1 using [3H]E1 as substrate by HPLC analysis | Homo sapiens | 9 | assay format | Scientific Literature | ||
| 5. | ALA1919077 | B | Selectivity ratio of IC50 for human placental cytosolic 17beta-HSD1 to IC50 for human placental microsomal 17beta-HSD2 | Homo sapiens | 9 | assay format | Scientific Literature | ||
| 6. | ALA1919078 | B | Displacement of [3H]E2 from human recombinant ERalpha by liquid scintillation counting relative to E2 | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 7. | ALA1919079 | B | Displacement of [3H]E2 from human recombinant ERbeta by liquid scintillation counting relative to E2 | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 8. | ALA1919080 | B | Inhibition of 17beta-HSD2 in human MDA-MB-231 cells after 3.5 hrs by HPLC analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 9. | ALA1919081 | B | Inhibition of human 17beta-HSD4 expressed in Escherichia coli assessed as radiolabeled E1 formation using [6,7-3H]E2 as substrate at 1 uM by scintillation counting | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA1919082 | B | Inhibition of human 17beta-HSD5 expressed in Escherichia coli assessed as radiolabeled testosterone formation using [1,2,6,7-3H]A-dione as substrate at 1 uM by scintillation counting | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA1919083 | B | Inhibition of human placental cytosolic 17beta-HSD2 assessed as inhibition of E1 formation using [2,4,6,7-3H]E2 as substrate at 1 uM after 20 mins by HPLC analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA1919084 | B | Inhibition of human placental cytosolic 17beta-HSD2 assessed as inhibition of E1 formation using [2,4,6,7-3H]E2 as substrate at 100 nM after 20 mins by HPLC analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA1919085 | B | Inhibition of human placental cytosolic 17beta-HSD1 assessed as inhibition of E2 formation using [2,4,6,7-3H]E1 as substrate at 1 uM after 10 mins by HPLC analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA1919086 | B | Inhibition of human placental cytosolic 17beta-HSD1 assessed as inhibition of E2 formation using [2,4,6,7-3H]E1 as substrate at 100 nM after 10 mins by HPLC analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA1919087 | B | Inhibition of rat liver microsomal 17beta-HSD2 assessed as inhibition of E1 formation using [2,4,6,7-3H]E2 as substrate at 1 uM after 20 mins by HPLC analysis | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 16. | ALA1919088 | B | Inhibition of rat liver microsomal 17beta-HSD1 assessed as inhibition of E2 formation using [2,4,6,7-3H]E1 as substrate at 1 uM after 10 mins by HPLC analysis | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 17. | ALA1919089 | B | Inhibition of mouse liver microsomal 17beta-HSD2 assessed as inhibition of E1 formation using [2,4,6,7-3H]E2 as substrate at 1 uM after 20 mins by HPLC analysis | Mus musculus | 1 | assay format | Scientific Literature | ||
| 18. | ALA1919139 | B | Inhibition of mouse liver microsomal 17beta-HSD1 assessed as inhibition of E2 formation using [2,4,6,7-3H]E1 as substrate at 1 uM after 10 mins by HPLC analysis | Mus musculus | 1 | assay format | Scientific Literature | ||
| 19. | ALA1919140 | B | Inhibition of monkey placental microsomal 17beta-HSD2 assessed as inhibition of E1 formation using [2,4,6,7-3H]E2 as substrate at 1 uM after 10 mins by HPLC analysis | Callithrix jacchus | 1 | assay format | Scientific Literature | ||
| 20. | ALA1919141 | B | Inhibition of monkey placental microsomal 17beta-HSD2 assessed as inhibition of E1 formation using [2,4,6,7-3H]E2 as substrate at 100 nM after 10 mins by HPLC analysis | Callithrix jacchus | 1 | assay format | Scientific Literature |
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