| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1936031 | B | Inhibition of human recombinant FAK expressed in baculovirus expression system after 30 mins by time resolved fluorescence assay | Homo sapiens | 21 | assay format | Scientific Literature | ||
| 2. | ALA1936085 | B | Inhibition of human recombinant JAK2 expressed in baculovirus expression system after 20 mins by time resolved fluorescence assay | Homo sapiens | 21 | assay format | Scientific Literature | ||
| 3. | ALA2161941 | F | Induction of apoptosis in ALK-dependent human SUP-M2 cells assessed as caspase 3/7 activation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA2161942 | B | Inhibition of GST-tagged human ALK cytoplasmic domain (1058-1620) expressed in Sf21 insect cells using GST-tagged human recombinant PLC-gamma/substrate by ELISA | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
| 5. | ALA2161943 | A | Half life in Sprague-Dawley rat liver microsomes at 0.5 uM preincubated for 10 mins before NADPH and UDPGA challenge | Rattus norvegicus | 13 | microsome format | Scientific Literature | ||
| 6. | ALA2161944 | A | Half life in monkey liver microsomes at 0.5 uM preincubated for 10 mins before NADPH and UDPGA challenge | Macaca mulatta | 10 | microsome format | Scientific Literature | ||
| 7. | ALA2161945 | A | Half life in human liver microsomes at 0.5 uM preincubated for 10 mins before NADPH and UDPGA challenge | Homo sapiens | 10 | microsome format | Scientific Literature | ||
| 8. | ALA2161946 | A | Half life in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 8 | organism-based format | Scientific Literature | ||
| 9. | ALA2161947 | A | Clearance in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 8 | organism-based format | Scientific Literature | ||
| 10. | ALA2161948 | A | Oral bioavailability in Sprague-Dawley rat at 5 mg/kg | Rattus norvegicus | 9 | organism-based format | Scientific Literature | ||
| 11. | ALA2161949 | B | Inhibition of IR | 12 | single protein format | Scientific Literature | |||
| 12. | ALA2161950 | A | AUC (0 to t) in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 13. | ALA2162253 | A | Volume of distribution in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 14. | ALA2162254 | A | Cmax in Sprague-Dawley rat at 5 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 15. | ALA2162255 | A | Tmax in Sprague-Dawley rat at 5 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 16. | ALA2162256 | A | AUC (0 to t) in Sprague-Dawley rat at 5 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 17. | ALA2162257 | A | Half life in SCID mouse at 1 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 18. | ALA2162258 | A | AUC (0 to t) in SCID mouse at 1 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 19. | ALA2162259 | A | Volume of distribution in SCID mouse at 1 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 20. | ALA2162260 | A | Clearance in SCID mouse at 1 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature |
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