| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1936672 | B | Displacement of [3H]histamine from human H4 receptor expressed in HEK cell membranes | Homo sapiens | 33 | cell-based format | Scientific Literature | ||
| 2. | ALA1936673 | A | Metabolic stability in human liver microsomes assessed as compound remaining after 60 mins | Homo sapiens | 1 | microsome format | Scientific Literature | ||
| 3. | ALA1936674 | A | Metabolic stability in mouse liver microsomes assessed as compound remaining after 60 mins | Mus musculus | 1 | microsome format | Scientific Literature | ||
| 4. | ALA1936675 | A | Metabolic stability in rat liver microsomes assessed as compound remaining after 60 mins | Rattus norvegicus | 1 | microsome format | Scientific Literature | ||
| 5. | ALA1936676 | A | Oral bioavailability in mouse | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 6. | ALA1936677 | A | Half life in mouse | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 7. | ALA1936678 | B | Displacement of [3H]histamine from human H3 receptor expressed in HEK cell membranes | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 8. | ALA1936679 | B | Displacement of [3H]histamine from human H1 receptor expressed in HEK cell membranes | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 9. | ALA1936680 | B | Displacement of cimetidine from H2 receptor at 10 uM | 4 | single protein format | Scientific Literature | |||
| 10. | ALA1936681 | F | Antagonist activity at human H4 receptor expressed in HEK293T cells assessed as inhibition of histamine-induced [35S]GTPgammaS binding | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 11. | ALA1936682 | B | Displacement of [3H]histamine from rat H1R | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 12. | ALA1936683 | B | Displacement of [3H]histamine from rat H3R | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 13. | ALA1936684 | B | Displacement of [3H]histamine from rat H4R | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 14. | ALA1936685 | B | Displacement of [3H]histamine from mouse H1R | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 15. | ALA1936686 | B | Displacement of [3H]histamine from mouse H3R | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 16. | ALA1936570 | B | Displacement of [3H]histamine from mouse H4R | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 17. | ALA1936571 | B | Displacement of [3H]histamine from human H4R assessed as binding half life | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 18. | ALA1936572 | B | Selectivity ratio of Ki for human H3 receptor to Ki for human H4 receptor | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA1936573 | B | Selectivity ratio of Ki for mouse H3 receptor to Ki for human H3 receptor | 1 | assay format | Scientific Literature | |||
| 20. | ALA1936574 | B | Selectivity ratio of Ki for rat H4 receptor to Ki for human H4 receptor | 1 | assay format | Scientific Literature |
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