| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1952467 | B | Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cells | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 2. | ALA1952468 | B | Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cells | Rattus norvegicus | 21 | cell-based format | Scientific Literature | ||
| 3. | ALA1952469 | F | Inverse agonist activity at human histamine H3 receptor assessed as inhibition of R-alpha-methylhistamine-induced [35S]GTPgammaS binding | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 4. | ALA1952470 | A | Apparent permeability across human Caco2 cells | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 5. | ALA1952473 | A | Half life in human liver microsomes | Homo sapiens | 2 | microsome format | Scientific Literature | ||
| 6. | ALA1952474 | A | Half life in rat liver microsomes | Rattus norvegicus | 2 | microsome format | Scientific Literature | ||
| 7. | ALA1952475 | A | Half life in dog liver microsomes | Canis lupus familiaris | 2 | microsome format | Scientific Literature | ||
| 8. | ALA1952476 | A | Half life in monkey liver microsomes | Macaca mulatta | 2 | microsome format | Scientific Literature | ||
| 9. | ALA1952477 | A | Inhibition of CYP1A2 | 2 | single protein format | Scientific Literature | |||
| 10. | ALA1952478 | A | Inhibition of CYP2C9 | 2 | single protein format | Scientific Literature | |||
| 11. | ALA1952479 | A | Inhibition of CYP2C19 | 2 | single protein format | Scientific Literature | |||
| 12. | ALA1952480 | A | Inhibition of CYP2D6 | 2 | single protein format | Scientific Literature | |||
| 13. | ALA1952481 | A | Inhibition of CYP3A4 | 2 | single protein format | Scientific Literature | |||
| 14. | ALA1952485 | B | Inhibition of DAT at 10 uM | 3 | single protein format | Scientific Literature | |||
| 15. | ALA1952486 | B | Inhibition of human Erg by patch clamp assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 16. | ALA1952487 | A | Half life in rat at 1 mg/kg, iv | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 17. | ALA1952488 | A | Volume of distribution in rat at 1 mg/kg, iv | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 18. | ALA1952489 | A | Clearance in rat at 1 mg/kg, iv | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 19. | ALA1952490 | A | Cmax in rat at 5 mg/kg, po | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 20. | ALA1952491 | A | Oral bioavailability in rat at 5 mg/kg | Rattus norvegicus | 4 | organism-based format | Scientific Literature |
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