| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2212446 | T | Toxicity in C57BL/6J mouse assessed as bloody stools at 150 mg/kg, po | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 2. | ALA2212447 | T | Toxicity in C57BL/6J mouse assessed as heavy breathing at 150 mg/kg, po after 1 to 4 hrs | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 3. | ALA2212448 | T | Toxicity in C57BL/6J mouse assessed as hunching at 150 mg/kg, po after 1 to 4 hrs | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 4. | ALA2212454 | A | Drug metabolism in C57Bl/6 mouse at 10 mg/kg, ip measured within 4 hrs by LC-MS/MS analysis | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 5. | ALA2212455 | A | Half life in mouse liver microsomes | Mus musculus | 2 | ALA2202988 | microsome format | Scientific Literature | |
| 6. | ALA2212456 | A | Drug metabolism in C57Bl/6 mouse at 10 mg/kg, iv measured within 2 hrs by LC-MS/MS analysis | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 7. | ALA2212458 | F | Induction of apoptosis in human MDA-MB-231 cells assessed as increase in caspase-3 activity | Homo sapiens | 2 | ALA2202988 | cell-based format | Scientific Literature | |
| 8. | ALA2212460 | F | Antiproliferative activity against human MDA-MB-231 cells assessed as Ki-67 level at 100 to 400 uM | Homo sapiens | 3 | ALA2202988 | cell-based format | Scientific Literature | |
| 9. | ALA2212462 | F | Cytotoxicity against human MDA-MB-231 cells assessed as decrease in cell number at 400 uM after 96 hrs by trypan blue assay | Homo sapiens | 3 | ALA2202988 | cell-based format | Scientific Literature | |
| 10. | ALA2212463 | F | Cytotoxicity against human MDA-MB-231 cells assessed as decrease in cell viability at 200 to 400 uM after 96 hrs by trypan blue assay | Homo sapiens | 2 | ALA2202988 | cell-based format | Scientific Literature | |
| 11. | ALA2212464 | T | Toxicity in po dosed C57BL/6J mouse | Mus musculus | 3 | ALA2202988 | organism-based format | Scientific Literature | |
| 12. | ALA2212466 | T | Toxicity in C57BL/6J mouse assessed as loss in body weight at 100 to 150 mg/kg, po after 96 hrs | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 13. | ALA2212467 | T | Toxicity in C57BL/6J mouse assessed as anxiety at 150 mg/kg, po after 1 to 4 hrs | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 14. | ALA2212468 | T | Toxicity in C57BL/6J mouse assessed as occurrence of diarrhea at 150 mg/kg, po after 2 to 3 days | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 15. | ALA2212469 | T | Toxicity in C57BL/6J mouse assessed as body shaking at 150 mg/kg, po after 1 to 4 hrs | Mus musculus | 1 | ALA2202988 | organism-based format | Scientific Literature | |
| 16. | ALA2212470 | B | Selectivity ratio of Kinact to Ki for PAD1 to Kinact to Ki for PAD4 | 6 | ALA2202988 | assay format | Scientific Literature | ||
| 17. | ALA2212471 | B | Selectivity ratio of Kinact to Ki for PAD1 to Kinact to Ki for PAD3 | 6 | ALA2202988 | assay format | Scientific Literature | ||
| 18. | ALA2212939 | B | Ratio of Kinact to Ki for PAD4 | 11 | ALA2202988 | single protein format | Scientific Literature | ||
| 19. | ALA2212940 | B | Selectivity ratio of Kinact to Ki for PAD1 to Kinact to Ki for PAD2 | 6 | ALA2202988 | assay format | Scientific Literature | ||
| 20. | ALA2212941 | B | Ratio of Kinact to Ki for PAD3 | 11 | ALA2202988 | single protein format | Scientific Literature |
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