# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3815885 | Binding | Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting method | Rattus norvegicus | 10 | ALA3813687 | cell-based format | Scientific Literature | |
2. | ALA645211 | Binding | Displacement of [3H]clonidine from rat cortex membrane Alpha-2 adrenergic receptors | Rattus norvegicus | 13 | ALA1144993 | assay format | Scientific Literature | |
3. | ALA641157 | Binding | Displacement of [3H]-clonidine from Alpha-2 adrenergic receptor of rat cortex membranes | Rattus norvegicus | 4 | ALA1132147 | cell membrane format | Scientific Literature | |
4. | ALA648724 | Binding | Binding affinity for rat alpha-2 adrenergic receptor from crude P2 membranes | Rattus norvegicus | 4 | ALA1147410 | assay format | Scientific Literature | |
5. | ALA698300 | Binding | Binding affinity for imidazoline receptor I-2 in rabbit kidney homogenate (relative to [3H]-Idazoxan radioligand) | Oryctolagus cuniculus | 119 | ALA1133017 | assay format | Scientific Literature | |
6. | ALA698301 | Binding | Relative binding to I2 and I1 imidazoline receptors (ratio of pKi) | 2 | ALA1132147 | assay format | Scientific Literature | ||
7. | ALA698302 | Binding | Relative binding to I2 imidazoline and alpha-2 adrenergic receptors (ratio of pKi) | 2 | ALA1132147 | assay format | Scientific Literature | ||
8. | ALA822086 | Functional | Compound was evaluated for hypotensive activity;no data | 5 | ALA1136789 | assay format | Scientific Literature | ||
9. | ALA841023 | Binding | Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranes | Rattus norvegicus | 1 | ALA1132147 | cell-based format | Scientific Literature | |
10. | ALA841024 | Binding | Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranes | Rattus norvegicus | 4 | ALA1132147 | cell-based format | Scientific Literature | |
11. | ALA841026 | Binding | Binding affinity for rat imidazoline receptor I-1 from crude P2 membranes | Rattus norvegicus | 4 | ALA1147410 | assay format | Scientific Literature | |
12. | ALA841027 | Binding | Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cells | Rattus norvegicus | 14 | ALA1144993 | cell-based format | Scientific Literature | |
13. | ALA842748 | Binding | Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | Oryctolagus cuniculus | 13 | ALA1144993 | assay format | Scientific Literature | |
14. | ALA842750 | Binding | Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranes | Oryctolagus cuniculus | 4 | ALA1132147 | assay format | Scientific Literature | |
15. | ALA842306 | Binding | Binding affinity for rat imidazoline I2 receptor from crude P2 membranes | Rattus norvegicus | 7 | ALA1147410 | assay format | Scientific Literature | |
16. | ALA845131 | Binding | Relative binding to imidazoline I1 and alpha-2 adrenergic receptors (ratio of pKi) | 13 | ALA1144993 | assay format | Scientific Literature | ||
17. | ALA845132 | Binding | Relative binding to imidazoline I1 and imidazoline I2 binding sites (ratio of pKi) | 13 | ALA1144993 | assay format | Scientific Literature | ||
18. | ALA663587 | Binding | Relative binding to imidazoline I2 and alpha-2 adrenergic receptors (ratio of pKi) | 13 | ALA1144993 | assay format | Scientific Literature | ||
19. | ALA717307 | Binding | Relative binding to imidazoline I2 and imidazoline I1 binding sites (ratio of pKi) | 13 | ALA1144993 | assay format | Scientific Literature | ||
20. | ALA839899 | Functional | Inhibition of MAO in rat liver assessed as inhibition of [14C]tyramine oxidation at 0.1 uM | Rattus norvegicus | 22 | ALA1146920 | assay format | Scientific Literature |