| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA643700 | B | Antilog of the difference between pD2 of Alpha-2 adrenergic receptor and pD2 of Alpha-1 adrenergic receptor | 8 | ALA1135400 | protein format | Scientific Literature | ||
| 2. | ALA643212 | F | Activation of recombinant human adrenergic, alpha-1D receptor expressed in rat-1 fibroblasts assayed via calcium mobilization through Gq coupled PLC pathway; No data. | 21 | ALA1135838 | assay format | Scientific Literature | ||
| 3. | ALA641224 | F | Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblasts; expressed as a percent of the maximal effect of the phenylephrine | 21 | ALA1134991 | assay format | Scientific Literature | ||
| 4. | ALA641225 | F | Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblasts | 23 | ALA1134991 | assay format | Scientific Literature | ||
| 5. | ALA641226 | B | In vitro binding affinity against cloned human alpha-1A-adrenoceptor receptors expressed in rat-1 fibroblasts | 8 | ALA1134991 | assay format | Scientific Literature | ||
| 6. | ALA641228 | F | Activation of human alpha-1B adrenergic receptors expressed in rat-1 fibroblasts | 23 | ALA1134991 | assay format | Scientific Literature | ||
| 7. | ALA641229 | B | In vitro binding affinity against cloned human alpha-1B-adrenoceptor receptors expressed in rat-1 fibroblasts | 8 | ALA1134991 | assay format | Scientific Literature | ||
| 8. | ALA641400 | F | Activation of human Alpha-1D adrenergic receptors expressed in rat-1 fibroblasts | 23 | ALA1134991 | assay format | Scientific Literature | ||
| 9. | ALA641401 | B | In vitro binding affinity against cloned human alpha-1D-adrenoceptor receptors expressed in rat-1 fibroblasts | 8 | ALA1134991 | assay format | Scientific Literature | ||
| 10. | ALA643412 | F | Activation of recombinant human adrenergic, alpha-1D receptor expressed in rat-1 fibroblasts assayed via calcium mobilization through Gq coupled PLC pathway | 30 | ALA1135838 | assay format | Scientific Literature | ||
| 11. | ALA643421 | B | Binding affinity of compound towards human Alpha-1D adrenergic receptor expressed in rat-1 fibroblast membranes | 6 | ALA1135838 | cell membrane format | Scientific Literature | ||
| 12. | ALA643027 | B | pD2 is -log ED50 required to produce 50% inhibition of the twitch response in rat vas deferens (intrinsic activity in presence of clonidine) for Alpha-2 adrenergic receptor | 6 | ALA1135400 | tissue-based format | Scientific Literature | ||
| 13. | ALA640225 | B | Displacement of [3H]clonidine from Alpha-2 adrenergic receptor of rat cortex membrane | Rattus norvegicus | 13 | ALA1135400 | assay format | Scientific Literature | |
| 14. | ALA643867 | B | Inhibition of Alpha-1 adrenergic receptor twitch response in rat vas deferens in presence of cirazoline, pD2 is -log ED50 | Rattus norvegicus | 12 | ALA1135400 | tissue-based format | Scientific Literature | |
| 15. | ALA649811 | B | Relative binding affinity for Alpha-2 adrenergic receptor and I2 imidazoline binding site (Antilog of the difference between pKi) | 13 | ALA1135400 | assay format | Scientific Literature | ||
| 16. | ALA647826 | F | Ability to activate cloned human alpha-1A receptor expressed in rat-1 fibroblasts via calcium mobilization through Gq coupled PLC pathway expressed as percent of phenylephrine (40 uM) response | 25 | ALA1135838 | assay format | Scientific Literature | ||
| 17. | ALA650229 | F | Activation of recombinant human adrenergic,alpha-1A receptor expressed in rat-1 fibroblasts determined via calcium mobilization through Gq coupled PLC pathway | 30 | ALA1135838 | assay format | Scientific Literature | ||
| 18. | ALA643738 | B | Binding affinity of compound towards Alpha-1A adrenergic receptor using membranes prepared from Rat-1 fibroblasts expressing human Alpha-1A adrenergic receptor | 6 | ALA1135838 | assay format | Scientific Literature | ||
| 19. | ALA652785 | F | Activation of human alpha-1B receptor expressed in rat-1 fibroblasts determined via calcium mobilization through Gq coupled PLC pathway expressed as percent of phenylephrine (40 um) response; No data | Homo sapiens | 18 | ALA1135838 | assay format | Scientific Literature | |
| 20. | ALA651230 | F | Activation of recombinant human adrenergic, alpha-1B receptor expressed in rat-1 fibroblasts determined via calcium mobilization through Gq coupled PLC pathway | 30 | ALA1135838 | assay format | Scientific Literature |
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