| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2014359 | B | Displacement of [3H]R-PIA from human recombinant adenosine receptor-1 expressed in CHO cell membrane after 60 mins by liquid scintillation counting | Homo sapiens | 19 | ALA2010736 | cell-based format | Scientific Literature | |
| 2. | ALA2014361 | B | Displacement of [3H]CGS21680 from human recombinant adenosine receptor-2A expressed in HEK293 cell membrane after 60 mins by liquid scintillation counting | Homo sapiens | 11 | ALA2010736 | cell-based format | Scientific Literature | |
| 3. | ALA2014402 | B | Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-counting | Homo sapiens | 22 | ALA2010736 | cell-based format | Scientific Literature | |
| 4. | ALA2014403 | F | Agonist activity at human recombinant adenosine receptor-1 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production at 10 uM preincubated for 45 mins prior forskolin-induction measured after 15 mins by immunoassay relative to 10 uM CPA | Homo sapiens | 15 | ALA2010736 | cell-based format | Scientific Literature | |
| 5. | ALA2014404 | F | Agonist activity at human recombinant adenosine receptor-1 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production preincubated for 45 mins prior forskolin-induction measured after 15 mins by immunoassay | Homo sapiens | 2 | ALA2010736 | cell-based format | Scientific Literature | |
| 6. | ALA2014405 | B | Displacement of [3H]R-PIA from rat forebrain adenosine receptor-1 | Rattus norvegicus | 8 | ALA2010736 | assay format | Scientific Literature | |
| 7. | ALA2014406 | B | Selectivity ratio of Ki for human recombinant adenosine receptor-3 to Ki for human recombinant adenosine receptor-1 | Homo sapiens | 5 | ALA2010736 | assay format | Scientific Literature | |
| 8. | ALA2014407 | B | Selectivity ratio of Ki for human recombinant adenosine receptor-2A to Ki for human recombinant adenosine receptor-1 | Homo sapiens | 2 | ALA2010736 | assay format | Scientific Literature | |
| 9. | ALA2173093 | B | Activity at human A2B adenosine receptor expressed in CHO cells assessed as stimulation of adenylate cyclase relative to control | Homo sapiens | 1 | ALA2169760 | cell-based format | Scientific Literature | |
| 10. | ALA2173094 | F | Anticonvulsant activity in CF-1 albino mouse assessed as protection against subcutaneous metrazol-induced seizures at 1 mg/kg, ip | Mus musculus | 3 | ALA2169760 | organism-based format | Scientific Literature | |
| 11. | ALA2173095 | F | Anticonvulsant activity in CF-1 albino mouse assessed as protection against subcutaneous metrazol-induced seizures at 3 mg/kg, ip | Mus musculus | 3 | ALA2169760 | organism-based format | Scientific Literature | |
| 12. | ALA2173096 | F | Anticonvulsant activity in CF-1 albino mouse assessed as protection against maximal electroshock-induced seizures at 2 mg/kg, ip by MES test | Mus musculus | 3 | ALA2169760 | organism-based format | Scientific Literature | |
| 13. | ALA2173097 | F | Anticonvulsant activity in CF-1 albino mouse assessed as protection against maximal electroshock-induced seizures at 1 mg/kg, ip by MES test | Mus musculus | 3 | ALA2169760 | organism-based format | Scientific Literature | |
| 14. | ALA2173098 | F | Anticonvulsant activity in CF-1 albino mouse assessed as protection against maximal electroshock-induced seizures at 3 mg/kg, ip by MES test | Mus musculus | 3 | ALA2169760 | organism-based format | Scientific Literature | |
| 15. | ALA2173099 | F | Anticonvulsant activity in ip dosed CF-1 albino mouse assessed as protection against 6 Hz psychomotor seizure after 1 hr by minimal clonic seizure test | Mus musculus | 3 | ALA2169760 | organism-based format | Scientific Literature | |
| 16. | ALA2173102 | T | Toxicity in ip dosed CF-1 albino mouse assessed as behavioral changes by rotarod test | Mus musculus | 1 | ALA2169760 | organism-based format | Scientific Literature | |
| 17. | ALA2174884 | F | Activity at human A1 adenosine receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production at 10 uM after 30 min | Homo sapiens | 26 | ALA2169760 | cell-based format | Scientific Literature | |
| 18. | ALA2174885 | B | Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cells after 60 min Packard Cobra 2 gamma-counter | Homo sapiens | 22 | ALA2169760 | cell-based format | Scientific Literature | |
| 19. | ALA2174887 | B | Displacement of [3H]CGS21680 from human A2a adenosine receptor expressed in HEK293 cells after 60 min by Perkin Elmer Liquid Scintillation Analyzer | Homo sapiens | 17 | ALA2169760 | cell-based format | Scientific Literature | |
| 20. | ALA2174889 | B | Displacement of [3H]R-PIA from human A1 adenosine receptor expressed in CHO cells after 60 min by Perkin Elmer Liquid Scintillation Analyzer | Homo sapiens | 23 | ALA2169760 | cell-based format | Scientific Literature |
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