| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2014888 | F | Antiinflammatory activity in rat RBL2H3 cells assessed as inhibition of DNP-BSA-induced TNF-alpha production preincubated for 15 mins prior DNP-BSA challenge measured after 30 mins by ELISA | Rattus norvegicus | 6 | ALA2010773 | cell-based format | Scientific Literature | |
| 2. | ALA2411915 | B | Inhibition of human USP5 using Ub-AMC as substrate at 1 to 20 uM after 10 mins by fluorometric analysis | Homo sapiens | 1 | ALA2406999 | single protein format | Scientific Literature | |
| 3. | ALA2411916 | B | Inhibition of human UCH-L1 using Ub-AMC as substrate at 1 to 20 uM after 10 mins by fluorometric analysis | Homo sapiens | 1 | ALA2406999 | single protein format | Scientific Literature | |
| 4. | ALA2411917 | B | Inhibition of human USP4 using Ub-AMC as substrate at 1 to 20 uM after 10 mins by fluorometric analysis | Homo sapiens | 1 | ALA2406999 | single protein format | Scientific Literature | |
| 5. | ALA2412074 | B | Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using K48-linked tetraubiquitin as substrate assessed as substrate hydrolysis at 20 uM after 15 mins by SDS-PAGE analysis | Homo sapiens | 1 | ALA2406999 | assay format | Scientific Literature | |
| 6. | ALA2412079 | B | Competitive binding affinity to human recombinant USP5 after 1 hr by SDS-PAGE analysis in presence of biotin-DMT | Homo sapiens | 2 | ALA2406999 | single protein format | Scientific Literature | |
| 7. | ALA4479671 | B | Inhibition of recombinant human 6His-tagged SENP1 catalytic domain expressed in Escherichia coli preincubated for 15 mins followed by addition of SUMO1-AMC as substrate measured after 1 hr by fluorescence analysis | Homo sapiens | 5 | ALA4477251 | assay format | Scientific Literature | |
| 8. | ALA4479672 | B | Inhibition of full-length recombinant human 6His-tagged SENP1 expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by addition of SUMO1-AMC as substrate measured after 1 hr by fluorescence analysis | Homo sapiens | 5 | ALA4477251 | assay format | Scientific Literature | |
| 9. | ALA4479675 | B | Inhibition of SENP1 in human KU812 cells preincubated for 20 mins followed by addition of HA-SUMO1-VS as substrate measured after 2 hrs by immunoblot analysis | Homo sapiens | 3 | ALA4477251 | cell-based format | Scientific Literature |
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