| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2026858 | F | Agonist activity at human alpha7 nAChR expressed in GH4C1 cells by FLIPR assay | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
| 2. | ALA2026859 | F | Agonist activity at human alpha7 nAChR expressed in GH4C1 cells by FLIPR assay relative to control | Homo sapiens | 24 | cell-based format | Scientific Literature | ||
| 3. | ALA2026860 | B | Displacement of [3H]Dofetilide from human ERG expressed in CHO-K1 cells by scintillation proximity assay | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
| 4. | ALA2026861 | A | Intrinsic permeability of the compound in MDCK cells expressing MDR1 | Canis lupus familiaris | 10 | cell-based format | Scientific Literature | ||
| 5. | ALA2026862 | A | Efflux ratio of intrinsic permeability of the compound in MDCK cells expressing MDR1 | Canis lupus familiaris | 9 | cell-based format | Scientific Literature | ||
| 6. | ALA2026863 | A | Clearance in rat liver assessed per gram of tissue | Rattus norvegicus | 3 | tissue-based format | Scientific Literature | ||
| 7. | ALA2026864 | A | Clearance in human liver assessed per gram of tissue | Homo sapiens | 3 | tissue-based format | Scientific Literature | ||
| 8. | ALA2026865 | B | Inhibition of human ERG | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA2026866 | A | Blood clearance in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 10. | ALA2026867 | A | Half life in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 11. | ALA2026868 | A | Tmax in Sprague-Dawley rat at 3 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 12. | ALA2026869 | A | Oral bioavailability in Sprague-Dawley rat at 3 mg/kg | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 13. | ALA2026871 | A | Ratio of drug level in brain to blood in CD1 mouse at 5 mg/kg, po after 3 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 14. | ALA2026872 | A | Inhibition of CYP1A2 | 1 | single protein format | Scientific Literature | |||
| 15. | ALA2026873 | A | Inhibition of CYP2C9 | 1 | single protein format | Scientific Literature | |||
| 16. | ALA2026874 | A | Inhibition of CYP2C19 | 1 | single protein format | Scientific Literature | |||
| 17. | ALA2026875 | A | Inhibition of CYP2D6 | 1 | single protein format | Scientific Literature | |||
| 18. | ALA2026876 | A | Inhibition of CYP3A4 using diethoxyfluorescein as substrate | 1 | single protein format | Scientific Literature | |||
| 19. | ALA2026877 | A | Inhibition of CYP3A4 using 7-benzyloxyquinoline as substrate | 1 | single protein format | Scientific Literature | |||
| 20. | ALA2026878 | F | Antagonist activity at alpha1 nAChR | 1 | assay format | Scientific Literature |
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