| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2025456 | Binding | Displacement of [I125]CGRP from CGRP receptor in human SK-N-MC cell membrane after 2 hrs by gamma or scintillation counting | Homo sapiens | 45 | ALA2021833 | cell-based format | Scientific Literature | |
| 2. | ALA2026482 | ADME | Permeability across human Caco2 cells | Homo sapiens | 13 | ALA2021833 | cell-based format | Scientific Literature | |
| 3. | ALA2026486 | Functional | Antagonist activity at CGRP receptor in human SK-N-MC cells assessed as inhibition of CGRP-stimulated cAMP production in presence of plasma | Homo sapiens | 2 | ALA2021833 | cell-based format | Scientific Literature | |
| 4. | ALA2026487 | ADME | Fraction unbound in po dosed rat plasma | Rattus norvegicus | 2 | ALA2021833 | organism-based format | Scientific Literature | |
| 5. | ALA2065547 | Functional | Antimigraine activity in marmosets assessed as inhibition of alphaCGRP-induced increase in facial blood flow at 10 mg/kg, po by laser Doppler flowmetry | marmosets | 1 | ALA2062501 | organism-based format | Scientific Literature | |
| 6. | ALA2065550 | Binding | Displacement of [125I]-CGRP from CGRP receptor in human SK-N-MC cells | Homo sapiens | 4 | ALA2062501 | cell-based format | Scientific Literature |
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