| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2025841 | B | Displacement of fluorescein-labeled phosphotyrosine-peptide derived from the interleukin-6 receptor subunit gp130 from the STAT3 after 15 mins by fluorescent polarization assay | 10 | single protein format | Scientific Literature | |||
| 2. | ALA2025842 | B | Displacement of 5-carboxyfluorescein-labeled GpYLVLDKW from the STAT5b-SH2 domain after 15 mins by fluorescent polarization assay | 10 | single protein format | Scientific Literature | |||
| 3. | ALA2025843 | B | Displacement of radioligand from the STAT1 after 15 mins by fluorescent polarization assay | 10 | single protein format | Scientific Literature | |||
| 4. | ALA2025844 | B | Selectivity ratio of Ki for STAT1 to Ki for STAT5b-SH2 domain | 6 | assay format | Scientific Literature | |||
| 5. | ALA2025845 | B | Selectivity ratio of Ki for STAT3 to Ki for STAT5b-SH2 domain | 6 | assay format | Scientific Literature | |||
| 6. | ALA2175186 | B | Inhibition of STAT3 SH2 domain assessed as inhibition of STAT3 SH2-phosphotyrosine interaction after 15 mins by fluorescence polarization assay | 6 | single protein format | Scientific Literature | |||
| 7. | ALA2175187 | B | Inhibition of STAT3 dimerization in v-Src transformed mouse NIH/3T3 cells overexpressing human EGFR assessed as suppression of STAT3-DNA interaction in nucleus after 30 mins by EMSA | Mus musculus | 12 | cell-based format | Scientific Literature |
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