| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2034300 | B | Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assay | Homo sapiens | 25 | ALA2029323 | single protein format | Scientific Literature | |
| 2. | ALA2034301 | B | Inhibition of human recombinant MAO-A assessed as H2O2 production by Resorufin/Amplex Red assay | Homo sapiens | 9 | ALA2029323 | single protein format | Scientific Literature | |
| 3. | ALA2034449 | B | Inhibition of human recombinant MAO-B assessed as H2O2 production by Resorufin/Amplex Red assay | Homo sapiens | 22 | ALA2029323 | single protein format | Scientific Literature | |
| 4. | ALA2034450 | B | Inhibition of human DAO measuring H2O2 production by Resorufin/Amplex Red assay | Homo sapiens | 5 | ALA2029323 | single protein format | Scientific Literature | |
| 5. | ALA2034551 | B | Inhibition of SSAO/VAP1 in mouse adipocytes measuring H2O2 production by Resorufin/Amplex Red assay | Mus musculus | 4 | ALA2029323 | cell-based format | Scientific Literature | |
| 6. | ALA2034552 | B | Selectivity ratio of IC50 for human MAO-B to IC50 for human SSAO/VAP1 | Homo sapiens | 3 | ALA2029323 | assay format | Scientific Literature | |
| 7. | ALA2034553 | B | Time dependent inhibition of human SSAO/VAP1 measuring H2O2 production by Resorufin/Amplex Red assay | Homo sapiens | 1 | ALA2029323 | single protein format | Scientific Literature | |
| 8. | ALA2034554 | B | Inhibition of human SSAO/VAP1 measuring H2O2 production by Kitz and Wilson plot analysis | Homo sapiens | 2 | ALA2029323 | single protein format | Scientific Literature | |
| 9. | ALA2034555 | B | Irreversible inhibition of human SSAO/VAP1 measuring H2O2 production after 24 hrs of dialysis by Resorufin/Amplex Red assay | Homo sapiens | 1 | ALA2029323 | single protein format | Scientific Literature | |
| 10. | ALA2034556 | T | Mutagenic activity in Salmonella typhimurium by Ames test | Salmonella enterica subsp. enterica serovar Typhimurium | 1 | ALA2029323 | organism-based format | Scientific Literature | |
| 11. | ALA2034557 | A | Inhibition of CYP450 | 1 | ALA2029323 | assay format | Scientific Literature | ||
| 12. | ALA2034558 | A | Oral bioavailability in rat | Rattus norvegicus | 1 | ALA2029323 | organism-based format | Scientific Literature | |
| 13. | ALA2034559 | A | Half life in po dosed rat | Rattus norvegicus | 1 | ALA2029323 | organism-based format | Scientific Literature | |
| 14. | ALA2034560 | F | Inhibition of SSAO/VAP1 in po dosed mouse gonadal adipose tissue after 6 hrs | Mus musculus | 1 | ALA2029323 | organism-based format | Scientific Literature | |
| 15. | ALA2034561 | F | Inhibition of SSAO/VAP1 in po dosed rat gonadal adipose tissue after 6 hrs | Rattus norvegicus | 1 | ALA2029323 | organism-based format | Scientific Literature | |
| 16. | ALA2034562 | F | Antiinflammatory activity in LPS-induced mouse assessed as decrease in cellular infiltration into BAL fluid at 100 mg/kg, ip administered 3 hrs prior LPS challenge relative to control | Mus musculus | 2 | ALA2029323 | organism-based format | Scientific Literature | |
| 17. | ALA2034563 | F | Antiinflammatory activity in LPS-induced mouse assessed as decrease in TNFalpha secretion at 100 mg/kg, ip administered 3 hrs prior LPS challenge relative to control | Mus musculus | 2 | ALA2029323 | organism-based format | Scientific Literature | |
| 18. | ALA2034564 | B | Inhibition of human AOC2 | Homo sapiens | 1 | ALA2029323 | single protein format | Scientific Literature |
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