| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2038472 | B | Displacement of 125I-MCP1 from human CCR2 receptor expressed in human THP-1 cell membrane by SPA assay | Homo sapiens | 38 | ALA2034889 | cell-based format | Scientific Literature | |
| 2. | ALA2038473 | F | Antagonist activity at human CCR2 receptor expressed in human THP-1 cells assessed as inhibition of MCP1-induced Ca2+ flux by FLIPR analysis | Homo sapiens | 38 | ALA2034889 | cell-based format | Scientific Literature | |
| 3. | ALA2038474 | B | Inhibition of human ERG | Homo sapiens | 38 | ALA2034889 | single protein format | Scientific Literature | |
| 4. | ALA2038485 | A | Intrinsic clearance in rat hepatocytes assessed per 10'6 cells | Rattus norvegicus | 2 | ALA2034889 | cell-based format | Scientific Literature | |
| 5. | ALA2038486 | A | Intrinsic clearance in dog hepatocytes assessed per 10'6 cells | Canis lupus familiaris | 1 | ALA2034889 | cell-based format | Scientific Literature | |
| 6. | ALA2038487 | A | Intrinsic clearance in human hepatocytes assessed per 10'6 cells | Homo sapiens | 1 | ALA2034889 | cell-based format | Scientific Literature | |
| 7. | ALA2038488 | A | Clearance in rat at 4 umol/kg, iv | Rattus norvegicus | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 8. | ALA2038489 | A | Clearance in dog at 4 umol/kg, iv | Canis lupus familiaris | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 9. | ALA2039170 | A | Volume of distribution at steady state in rat at 4 umol/kg, iv | Rattus norvegicus | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 10. | ALA2039622 | A | Volume of distribution at steady state in dog at 4 umol/kg, iv | Canis lupus familiaris | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 11. | ALA2039623 | A | Half life in rat at 4 umol/kg, iv | Rattus norvegicus | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 12. | ALA2039624 | A | Half life in dog at 4 umol/kg, iv | Canis lupus familiaris | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 13. | ALA2039625 | A | Oral bioavailability in rat at 11 umol/kg | Rattus norvegicus | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 14. | ALA2039626 | A | Oral bioavailability in dog at 4 umol/kg | Canis lupus familiaris | 1 | ALA2034889 | organism-based format | Scientific Literature | |
| 15. | ALA2039627 | P | Lipophilicity, log D of the compound at pH 7.4 | 2 | ALA2034889 | small-molecule physicochemical format | Scientific Literature | ||
| 16. | ALA2039628 | P | Lipophilicity, log P of the compound at pH 7.4 | 2 | ALA2034889 | small-molecule physicochemical format | Scientific Literature | ||
| 17. | ALA2039629 | P | Dissociation constant, pKa of the compound | 2 | ALA2034889 | small-molecule physicochemical format | Scientific Literature | ||
| 18. | ALA2039630 | P | Aqueous solubility of the compound | 1 | ALA2034889 | small-molecule physicochemical format | Scientific Literature | ||
| 19. | ALA2039631 | B | Inhibition of human ERG by electrophysiology assay | Homo sapiens | 1 | ALA2034889 | single protein format | Scientific Literature | |
| 20. | ALA2039632 | B | Selectivity ratio of IC50 for human ERG to IC50 for human CCR2 | Homo sapiens | 1 | ALA2034889 | assay format | Scientific Literature |
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