Assay

#	Aladdin ID	Assay Type	Description	Organism	Compounds	BAO Format	Source
1.	ALA2039222	B	Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assay		41	single protein format	Scientific Literature
2.	ALA2039223	B	Inhibition of RGS8 interaction with Galpha0 protein by flow cytometry protein interaction assay		41	single protein format	Scientific Literature
3.	ALA2039224	B	Selectivity ratio of IC50 for RGS8 to IC50 RGS4		40	assay format	Scientific Literature
4.	ALA3706279	B	Inhibitory Assay: FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyplex high throughput screen to identify inhibitors of the RGS-Gα interaction [4]. This activity was confirmed by analyzing the effect of CCG-50014 on several different RGS proteins with freshly reordered compound using multiplexed FCPIA. CCG-50014 fully inhibited several different RGS proteins including RGS4, 8, 16, and 19, but did not have activity on RGS7 or a mutated form of RGS4 that lacks cysteine residues.		4	single protein format	BindingDB Database
5.	ALA3707997	B	Inhibitory Assay: FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyplex high throughput screen to identify inhibitors of the RGS-Gα interaction [4]. This activity was confirmed by analyzing the effect of CCG-50014 on several different RGS proteins with freshly reordered compound using multiplexed FCPIA. CCG-50014 fully inhibited several different RGS proteins including RGS4, 8, 16, and 19, but did not have activity on RGS7 or a mutated form of RGS4 that lacks cysteine residues.	Homo sapiens	4	single protein format	BindingDB Database