| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2050764 | B | Ratio of Kinact to Ki for rat recombinant KAT2 using L-kynurenine as substrate | Rattus norvegicus | 8 | single protein format | Scientific Literature | ||
| 2. | ALA2050765 | B | Ratio of Kinact to Ki for human recombinant KAT2 using L-kynurenine as substrate | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 3. | ALA2050766 | B | Inhibition of human recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrs | Homo sapiens | 22 | single protein format | Scientific Literature | ||
| 4. | ALA2050767 | B | Inhibition of rat recombinant KAT2 assessed as conversion of L-kynurenine into kynurenic acid after 15 to 20 hrs | Rattus norvegicus | 21 | single protein format | Scientific Literature | ||
| 5. | ALA2329098 | B | Binding affinity to C-terminal hexa histidine tagged full length human KAT2 K240S/F241G mutant harboring C-terminal thrombin cleavage site at 1 mM after 2 hrs by X-ray crystallography in presence of 2 mM PLP | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 6. | ALA2329101 | B | Ratio of Kinact to Ki for rat KAT2 using L-kynurenine as substrate by SpectraMax plate reader analysis | Rattus norvegicus | 4 | single protein format | Scientific Literature | ||
| 7. | ALA2329105 | B | Inhibition of human KAT3 using L-kynurenine as substrate measured after 24 hrs by SpectraMax plate reader analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 8. | ALA2329107 | B | Ratio of Kinact to Ki for human KAT2 using L-kynurenine as substrate by SpectraMax plate reader analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 9. | ALA2329108 | B | Inhibition of human KAT1 using L-kynurenine as substrate measured after 16 hrs by SpectraMax plate reader analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 10. | ALA2329109 | B | Irreversible inhibition of human KAT2 using L-kynurenine as substrate measured every 5 mins over 16 hrs by SpectraMax plate reader analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 11. | ALA2329110 | B | Inhibition of human KAT2 using L-kynurenine as substrate measured after 15-20 hrs by SpectraMax plate reader analysis | Homo sapiens | 4 | single protein format | Scientific Literature |
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