| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2072750 | B | Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 2. | ALA2072751 | B | Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 3. | ALA2072752 | B | Inhibition of human ERG expressed in CHO cells by IonWorks HT assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 4. | ALA2072753 | P | Solubility of the compound | 31 | small-molecule physicochemical format | Scientific Literature | |||
| 5. | ALA2072754 | A | Intrinsic clearance in rat liver microsomes assessed per ug of protein | Rattus norvegicus | 31 | microsome format | Scientific Literature | ||
| 6. | ALA2072755 | A | Intrinsic clearance in human liver microsomes assessed per ug of protein | Homo sapiens | 31 | microsome format | Scientific Literature | ||
| 7. | ALA2072756 | B | Activity at 5HT receptor | Homo sapiens | 3 | protein format | Scientific Literature | ||
| 8. | ALA2072757 | A | Dose normalized AUC in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 9. | ALA2072758 | A | Volume of distribution at steady state in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 10. | ALA2072759 | A | Half life in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 11. | ALA2072760 | A | Clearance in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 12. | ALA2072761 | A | Dose normalized AUC in Sprague-Dawley rat at 10 umol/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 13. | ALA2072762 | A | Cmax in Sprague-Dawley rat at 10 umol/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 14. | ALA2072763 | A | Tmax in Sprague-Dawley rat at 10 umol/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 15. | ALA2072764 | A | Half life in Sprague-Dawley rat at 10 umol/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 16. | ALA2072765 | A | Oral bioavailability in Sprague-Dawley rat at 10 umol/kg | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 17. | ALA2072766 | B | Displacement of [3H]rauwolscine from adrenergic alpha2B receptor at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA2072767 | B | Displacement of [125I]RTI-55 from DAT at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA2072768 | B | Displacement of [125I]ghrelin from GHS receptor at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA2072769 | B | Displacement of [125I]RTI-55 from DAT | Homo sapiens | 1 | single protein format | Scientific Literature |
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