# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2072491 | B | Displacement of [35S]MK499 from human Erg expressed in HEK293 cells after 60 mins by scintillation counting | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
2. | ALA2072502 | B | Binding affinity to L-type calcium channel | Homo sapiens | 4 | assay format | Scientific Literature | ||
3. | ALA2072503 | A | Dose normalized AUC in C57BL/6N mouse at 2 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
4. | ALA2072504 | A | Cmax in C57BL/6N mouse at 2 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
5. | ALA2072505 | A | Volume of distribution at steady state in C57BL/6N mouse at 1 mg/kg, iv and 2 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
6. | ALA2072506 | A | Clearance in C57BL/6N mouse at 1 mg/kg, iv and 2 mg/kg, po | Mus musculus | 4 | organism-based format | Scientific Literature | ||
7. | ALA2072507 | A | Half life in C57BL/6N mouse at 1 mg/kg, iv and 2 mg/kg, po | Mus musculus | 3 | organism-based format | Scientific Literature | ||
8. | ALA2072508 | A | Oral bioavailability in C57BL/6N mouse at 2 mg/kg | Mus musculus | 3 | organism-based format | Scientific Literature | ||
9. | ALA2072627 | B | Selectivity for human SST3 receptor over human SST1 receptor | Homo sapiens | 3 | assay format | Scientific Literature | ||
10. | ALA2072628 | B | Selectivity for human SST3 receptor over human SST2 receptor | Homo sapiens | 3 | assay format | Scientific Literature | ||
11. | ALA2072629 | B | Selectivity for human SST3 receptor over human SST4 receptor | Homo sapiens | 3 | assay format | Scientific Literature | ||
12. | ALA2072630 | B | Selectivity for human SST3 receptor over human SST5 receptor | Homo sapiens | 3 | assay format | Scientific Literature | ||
13. | ALA2072631 | F | Antagonist activity at human SST3 receptor | Homo sapiens | 1 | assay format | Scientific Literature |