| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2072489 | B | Displacement of [125I]SS-14 from human SST3 receptor expressed in CHO cells after 60 mins by scintillation counting | Homo sapiens | 13 | ALA2069262 | cell-based format | Scientific Literature | |
| 2. | ALA2072490 | F | Antagonist activity at human SST3 receptor expressed in CHO cells assessed as inhibition of forskolin/SS-14-stimulated cAMP accumulation preincubated for 15 mins before SS-14 challenge measured after 1 hr by time-resolved fluorescence analysis | Homo sapiens | 12 | ALA2069262 | cell-based format | Scientific Literature | |
| 3. | ALA2072491 | B | Displacement of [35S]MK499 from human Erg expressed in HEK293 cells after 60 mins by scintillation counting | Homo sapiens | 14 | ALA2069262 | cell-based format | Scientific Literature | |
| 4. | ALA2072492 | B | Binding affinity to human SST1 receptor expressed in CHO cells | Homo sapiens | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 5. | ALA2072493 | B | Binding affinity to human SST2 receptor expressed in CHO cells | Homo sapiens | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 6. | ALA2072494 | B | Binding affinity to human SST4 receptor expressed in CHO cells | Homo sapiens | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 7. | ALA2072495 | B | Binding affinity to human SST5 receptor expressed in CHO cells | Homo sapiens | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 8. | ALA2072496 | B | Displacement of [125I]SS-14 from mouse SST3 receptor expressed in CHO cells after 60 mins by scintillation counting | Mus musculus | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 9. | ALA2072497 | F | Antagonist activity at mouse SST3 receptor expressed in CHO cells assessed as inhibition of forskolin/SS-14-stimulated cAMP accumulation preincubated for 15 mins before SS-14 challenge measured after 1 hr by time-resolved fluorescence analysis | Mus musculus | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 10. | ALA2072498 | B | Binding affinity to mouse SST1 receptor expressed in CHO cells | Mus musculus | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 11. | ALA2072499 | B | Binding affinity to mouse SST2 receptor expressed in CHO cells | Mus musculus | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 12. | ALA2072500 | B | Binding affinity to mouse SST4 receptor expressed in CHO cells | Mus musculus | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 13. | ALA2072501 | B | Binding affinity to mouse SST5 receptor expressed in CHO cells | Mus musculus | 1 | ALA2069262 | cell-based format | Scientific Literature | |
| 14. | ALA2072502 | B | Binding affinity to L-type calcium channel | Homo sapiens | 4 | ALA2069262 | assay format | Scientific Literature | |
| 15. | ALA2072503 | A | Dose normalized AUC in C57BL/6N mouse at 2 mg/kg, po | Mus musculus | 3 | ALA2069262 | organism-based format | Scientific Literature | |
| 16. | ALA2072504 | A | Cmax in C57BL/6N mouse at 2 mg/kg, po | Mus musculus | 3 | ALA2069262 | organism-based format | Scientific Literature | |
| 17. | ALA2072505 | A | Volume of distribution at steady state in C57BL/6N mouse at 1 mg/kg, iv and 2 mg/kg, po | Mus musculus | 3 | ALA2069262 | organism-based format | Scientific Literature | |
| 18. | ALA2072506 | A | Clearance in C57BL/6N mouse at 1 mg/kg, iv and 2 mg/kg, po | Mus musculus | 4 | ALA2069262 | organism-based format | Scientific Literature | |
| 19. | ALA2072507 | A | Half life in C57BL/6N mouse at 1 mg/kg, iv and 2 mg/kg, po | Mus musculus | 3 | ALA2069262 | organism-based format | Scientific Literature | |
| 20. | ALA2072508 | A | Oral bioavailability in C57BL/6N mouse at 2 mg/kg | Mus musculus | 3 | ALA2069262 | organism-based format | Scientific Literature |
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