| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2073576 | B | Inhibition of mouse PDE10A-mediated hydrolysis of [3H]cGMP to [3H]GMP after 20 mins by scintillation counting | Mus musculus | 49 | ALA2069174 | single protein format | Scientific Literature | |
| 2. | ALA2073577 | P | Metabolic stability of the compound in simulated gastric fluid | 2 | ALA2069174 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA2073578 | A | Oral bioavailability in mouse | Mus musculus | 2 | ALA2069174 | organism-based format | Scientific Literature | |
| 4. | ALA2073579 | A | Ratio of drug level in brain to plasma in mouse | Mus musculus | 2 | ALA2069174 | organism-based format | Scientific Literature | |
| 5. | ALA2073580 | B | Selectivity ratio for PDE1A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 6. | ALA2073581 | B | Selectivity ratio for PDE2A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 7. | ALA2073582 | B | Selectivity ratio for PDE3A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 8. | ALA2073583 | B | Selectivity ratio for PDE4A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 9. | ALA2073584 | B | Selectivity ratio for PDE5A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 10. | ALA2073585 | B | Selectivity ratio for PDE7A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 11. | ALA2073586 | B | Selectivity ratio for PDE8A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 12. | ALA2073587 | B | Selectivity ratio for PDE9A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 13. | ALA2073588 | B | Selectivity ratio for PDE11A to mouse PDE10A | 2 | ALA2069174 | assay format | Scientific Literature | ||
| 14. | ALA2073589 | F | Antipsychotic activity in mouse assessed as conditioned avoidance response at 10 mg/kg, po | Mus musculus | 2 | ALA2069174 | organism-based format | Scientific Literature | |
| 15. | ALA2073590 | F | Antipsychotic activity in mouse assessed as conditioned avoidance response at 5 mg/kg, po | Mus musculus | 2 | ALA2069174 | organism-based format | Scientific Literature | |
| 16. | ALA2073591 | F | Antipsychotic activity in mouse assessed as reduction of phencyclidine-induced hyperlocomotion at 4 to 5 mg/kg, po | Mus musculus | 1 | ALA2069174 | organism-based format | Scientific Literature | |
| 17. | ALA2073592 | F | Antipsychotic activity in mouse assessed as apparent memory restoration at 4 mg/kg, ip by object recognition assay | Mus musculus | 1 | ALA2069174 | organism-based format | Scientific Literature |
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