| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2073525 | B | Inhibition of IKKbeta using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins prior to substrate addition by IMAP-TR-FRET assay | Homo sapiens | 19 | single protein format | Scientific Literature | ||
| 2. | ALA2073526 | B | Inhibition of IKKbeta in human HeLa cells assessed as inhibition of TPA-induced NFkappaB activation at 10 uM incubated for 1 hr prior to TPA-challenge measured after 8 hrs by luciferase reporter gene assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 3. | ALA2073527 | B | Inhibition of IKKbeta in mouse CIA model splenocytes assessed as inhibition of TNFalpha production after 72 hrs by ELISA | Mus musculus | 14 | cell-based format | Scientific Literature | ||
| 4. | ALA2073528 | B | Inhibition of IKKalpha | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 5. | ALA2073529 | B | Inhibition of MAPK p38alpha | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA2073530 | B | Inhibition of MAPK p38beta | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 7. | ALA2073531 | B | Inhibition of JNK1 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 8. | ALA2073532 | B | Inhibition of JNK2 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA2073533 | B | Inhibition of JNK3 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 10. | ALA2073534 | B | Selectivity ratio of IC50 for IKKalpha to IC50 for IKKbeta | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 11. | ALA2073535 | B | Inhibition of IKKbeta using 5FAM-GRHDSGLDSMK-NH2 as substrate at 10 uM incubated for 10 mins prior to substrate addition by IMAP-TR-FRET assay | Homo sapiens | 31 | single protein format | Scientific Literature |
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