| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2092081 | B | Inhibition of PI3Kalpha in human U2OS cells assessed as inhibition of AKT Ser 473 phosphorylation by Western blot | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 2. | ALA2092082 | B | Inhibition of human PI3Kalpha (p110alpha/p85alpha) by ADP accumulation based HTRF assay | Homo sapiens | 36 | protein complex format | Scientific Literature | ||
| 3. | ALA2092083 | A | Stability in human liver microsomes at 1 uM incubated for 15 mins | Homo sapiens | 9 | microsome format | Scientific Literature | ||
| 4. | ALA2092084 | A | Stability in mouse liver microsomes at 1 uM incubated for 15 mins | Mus musculus | 9 | microsome format | Scientific Literature | ||
| 5. | ALA2092085 | A | Inhibition of CYP1A2 at 10 uM | 9 | single protein format | Scientific Literature | |||
| 6. | ALA2092086 | A | Inhibition of CYP2C9 at 10 uM | 9 | single protein format | Scientific Literature | |||
| 7. | ALA2092087 | A | Inhibition of CYP2C19 at 10 uM | 9 | single protein format | Scientific Literature | |||
| 8. | ALA2092088 | A | Inhibition of CYP2D6 at 10 uM | 9 | single protein format | Scientific Literature | |||
| 9. | ALA2092089 | A | Inhibition of CYP3A4 at 10 uM | 9 | single protein format | Scientific Literature | |||
| 10. | ALA2092090 | B | Inhibition of human PI3Kbeta (p110beta/p85alpha) by ADP accumulation based HTRF assay | Homo sapiens | 5 | protein complex format | Scientific Literature | ||
| 11. | ALA2092091 | B | Inhibition of human PI3Kdelta (p110delta/p85alpha) by ADP accumulation based HTRF assay | Homo sapiens | 5 | protein complex format | Scientific Literature | ||
| 12. | ALA2092092 | B | Inhibition of mTOR | 9 | single protein format | Scientific Literature | |||
| 13. | ALA2092093 | B | Inhibition of human PI3Kgamma by ADP accumulation based HTRF assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 14. | ALA2092094 | B | Inhibition of human PI3Kalpha E542K mutant by ADP accumulation based HTRF assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 15. | ALA2092095 | B | Inhibition of human PI3Kalpha E545K mutant by ADP accumulation based HTRF assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 16. | ALA2092096 | B | Inhibition of human PI3Kalpha H1047R mutant by ADP accumulation based HTRF assay | Homo sapiens | 5 | single protein format | Scientific Literature |
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