| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA874428 | B | Maximum percent of enhancement of binding. | 31 | ALA1123034 | protein complex format | Scientific Literature | ||
| 2. | ALA636847 | B | Compounds was evaluated for their ability to enhance (+/-)-[3H]nicotine binding at a particular dose range 5E-9 - 1.5E-8 was reported | 1 | ALA1123034 | protein complex format | Scientific Literature | ||
| 3. | ALA754768 | A | Inhibitory constant for cytochrome P450 2D6 | Homo sapiens | 6 | ALA1126649 | single protein format | Scientific Literature | |
| 4. | ALA909735 | B | Inhibition of [3H]NIC binding to alpha-4-beta-2 nAChR in rat brain membrane | Rattus norvegicus | 9 | ALA1149505 | cell membrane format | Scientific Literature | |
| 5. | ALA909736 | B | Inhibition of [3H]MLA binding to alpha-7 nAChR in rat brain membrane | Rattus norvegicus | 9 | ALA1149505 | cell membrane format | Scientific Literature | |
| 6. | ALA909737 | B | Inhibition of [3H]DA uptake at DAT in rat striatal synaptosomes | Rattus norvegicus | 9 | ALA1149505 | subcellular format | Scientific Literature | |
| 7. | ALA909738 | B | Inhibition of [3H]5-HT uptake at SERT in rat hippocampal synaptosomes | Rattus norvegicus | 9 | ALA1149505 | subcellular format | Scientific Literature | |
| 8. | ALA909739 | B | Inhibition of [3H]DTBZ binding to VMAT2 in rat synaptic vesicle membrane | Rattus norvegicus | 10 | ALA1149505 | cell membrane format | Scientific Literature | |
| 9. | ALA909740 | B | Selectivity for VMAT2 over DAT | Rattus norvegicus | 1 | ALA1149505 | assay format | Scientific Literature | |
| 10. | ALA909741 | B | Selectivity for VMAT2 over SERT | Rattus norvegicus | 1 | ALA1149505 | assay format | Scientific Literature | |
| 11. | ALA1047523 | B | Displacement of [3H]DTBZ from VMAT2 dihydrotetrabenazine binding site in rat brain synaptic vesicle by scintillation counting | Rattus norvegicus | 20 | ALA1155179 | tissue-based format | Scientific Literature | |
| 12. | ALA1047524 | B | Inhibition of [3H]dopamine uptake at VMAT2 in rat brain synaptic vesicle by liquid scintillation spectroscopy | Rattus norvegicus | 20 | ALA1155179 | tissue-based format | Scientific Literature | |
| 13. | ALA1047525 | B | Ratio of Ki for displacement of [3H]DTBZ from VMAT2 dihydrotetrabenazine binding site in rat brain synaptic vesicle to Ki for inhibition of [3H]dopamine uptake at VMAT2 in rat brain synaptic vesicle | Rattus norvegicus | 20 | ALA1155179 | tissue-based format | Scientific Literature | |
| 14. | ALA1068115 | B | Displacement of [3H]MLA from alpha7 nAChR in rat brain homogenate by liquid scintillation spectrophotometry | Rattus norvegicus | 21 | ALA1159052 | tissue-based format | Scientific Literature | |
| 15. | ALA1068116 | B | Displacement of [3H]nicotine from alpha4beta2 nAChR in rat brain homogenate by liquid scintillation spectrophotometry | Rattus norvegicus | 21 | ALA1159052 | tissue-based format | Scientific Literature | |
| 16. | ALA1068119 | B | Inhibition of [3H]DA uptake at DAT in rat brain striatal synaptosomes by liquid scintillation spectrophotometry | Rattus norvegicus | 22 | ALA1159052 | subcellular format | Scientific Literature | |
| 17. | ALA1068120 | B | Inhibition of [3H]5HT uptake at SERT in rat brain hippocampal synaptosomes by liquid scintillation spectrophotometry | Rattus norvegicus | 22 | ALA1159052 | subcellular format | Scientific Literature | |
| 18. | ALA1068123 | B | Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometry | Rattus norvegicus | 10 | ALA1159052 | assay format | Scientific Literature | |
| 19. | ALA1068126 | B | Selectivity ratio of Ki for rat VMAT2 to Ki for rat alpha4beta2 nAChR | Rattus norvegicus | 1 | ALA1159052 | assay format | Scientific Literature | |
| 20. | ALA1068127 | B | Binding affinity to VMAT2 receptor | 5 | ALA1159052 | single protein format | Scientific Literature |
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