| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3598911 | F | Antitrypanosomal activity against Trypanosoma brucei brucei 427 assessed as inhibition of parasite proliferation measured as ATP levels after 48 hrs by luciferase-based assay | Trypanosoma brucei brucei | 14 | organism-based format | Scientific Literature | ||
| 2. | ALA3598912 | B | Inhibition of human HDAC1 | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 3. | ALA3598913 | B | Inhibition of human HDAC2 | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 4. | ALA3598914 | B | Inhibition of human HDAC3 | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 5. | ALA3598915 | B | Inhibition of human HDAC8 | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 6. | ALA3598916 | B | Inhibition of human HDAC4 | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 7. | ALA3598917 | B | Inhibition of human HDAC5 | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 8. | ALA3598918 | B | Inhibition of human HDAC7 | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 9. | ALA3598919 | B | Inhibition of human HDAC9 | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 10. | ALA3598920 | B | Inhibition of human HDAC6 | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 11. | ALA3598921 | B | Inhibition of human HDAC10 | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 12. | ALA3598922 | B | Inhibition of human HDAC11 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 13. | ALA3598923 | A | Cmax in po dosed human measured under phase 1 trial | Homo sapiens | 5 | organism-based format | Scientific Literature | ||
| 14. | ALA3598927 | A | AUC in po dosed human measured under phase 1 trial | Homo sapiens | 5 | organism-based format | Scientific Literature | ||
| 15. | ALA3598931 | A | Tmax in po dosed human measured under phase 1 trial | Homo sapiens | 5 | organism-based format | Scientific Literature | ||
| 16. | ALA3860984 | A | Inhibition of full length recombinant human HDAC1 expressed in baculovirus infected Sf9 cells using RHKK-Ac as substrate by fluorescence analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA3860985 | A | Inhibition of full length recombinant human HDAC2 expressed in baculovirus infected Sf9 cells using RHKK-Ac as substrate by fluorescence analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA3860986 | A | Inhibition of full length recombinant human HDAC3/NCOR2 expressed in baculovirus infected Sf9 cells using RHKK-Ac as substrate by fluorescence analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA3860987 | B | Inhibition of full length recombinant human HDAC6 expressed in baculovirus infected Sf9 cells using RHKK-Ac as substrate by fluorescence analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA4009226 | A | Inhibition of recombinant human LTA4H aminopeptidase activity expressed in Escherichia coli BL21 (DE3) pLysS assessed as formation of p-NA from Ala-p-NA preincubated for 10 mins followed by substrate addition measured after 10 mins | Homo sapiens | 18 | assay format | Scientific Literature |
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