#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA2148460	B	Displacement of [Phe13, [125I]Tyr19]-MCH from human MCHR1 receptor E4Q/A5T mutant expressed in HEK 293 cell membranes by scintillation counter	Homo sapiens	2	ALA2146433	cell-based format	Scientific Literature
2.	ALA3858580	B	Displacement of [Phe13,125I]Tyr19]-MCH from human MCHR1 E4Q/A5T double mutant expressed in HEK293 cells by TopCount scintillation counting method	Homo sapiens	8	ALA3856239	cell-based format	Scientific Literature
3.	ALA3858581	A	Metabolic stability in human liver microsomes assessed as compound remaining at 3 uM measured after 10 min	Homo sapiens	7	ALA3856239	tissue-based format	Scientific Literature
4.	ALA3858582	A	Metabolic stability in rat liver microsomes assessed as compound remaining at 3 uM measured after 10 min	Rattus norvegicus	7	ALA3856239	tissue-based format	Scientific Literature
5.	ALA3858583	A	Metabolic stability in mouse liver microsomes assessed as compound remaining at 3 uM measured after 10 min	Mus musculus	7	ALA3856239	tissue-based format	Scientific Literature
6.	ALA3858584	P	Solubility of the compound in phosphate buffer at pH 6.4		13	ALA3856239	small-molecule physicochemical format	Scientific Literature
7.	ALA3858585	P	Lipophilicity, log P of the compound at pH 7 by HPLC analysis		7	ALA3856239	small-molecule physicochemical format	Scientific Literature
8.	ALA3858586	A	Protein binding in rat plasma assessed as unbound fraction	Rattus norvegicus	7	ALA3856239	cell-free format	Scientific Literature
9.	ALA3858591	T	Toxicity in DIO Sprague-Dawley rat assessed as biliary lesion formation at 10 mg/kg, po qd for 4 days	Rattus norvegicus	1	ALA3856239	organism-based format	Scientific Literature
10.	ALA3858596	B	Inhibition of MCHR2 (unknown origin) up to 10 uM	Homo sapiens	1	ALA3856239	single protein format	Scientific Literature
11.	ALA3858597	A	Protein binding in Sprague-Dawley rat plasma at 10 mg/kg, po qd for 4 days	Rattus norvegicus	6	ALA3856239	organism-based format	Scientific Literature
12.	ALA3858604	F	Antiobesity activity in pair-fed DIO Sprague-Dawley rat model assessed as reduction in body weight at 1 mg/kg, po qd for 28 days relative to vehicle control	Rattus norvegicus	1	ALA3856239	organism-based format	Scientific Literature
13.	ALA3858605	F	Antiobesity activity in pair-fed DIO Sprague-Dawley rat model assessed as reduction in body weight at 3 mg/kg, po qd for 28 days relative to vehicle control	Rattus norvegicus	1	ALA3856239	organism-based format	Scientific Literature
14.	ALA3858613	F	Antiobesity activity in pair-fed DIO Sprague-Dawley rat model assessed as reduction in caloric intake at 1 mg/kg, po qd for 28 days relative to vehicle control	Rattus norvegicus	1	ALA3856239	organism-based format	Scientific Literature
15.	ALA3858614	F	Antiobesity activity in pair-fed DIO Sprague-Dawley rat model assessed as reduction in caloric intake at 3 mg/kg, po qd for 28 days relative to vehicle control	Rattus norvegicus	1	ALA3856239	organism-based format	Scientific Literature
16.	ALA3858622	F	Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as inhibition of MCH-stimulated calcium flux measured after 15 mins by FLIPR assay	Homo sapiens	1	ALA3856239	cell-based format	Scientific Literature
17.	ALA3858623	F	Antagonist activity at human MCHR2 expressed in HEK293 cells assessed as inhibition of MCH-stimulated calcium flux at 10 uM measured after 15 mins by FLIPR assay	Homo sapiens	1	ALA3856239	cell-based format	Scientific Literature
18.	ALA3858624	B	Binding affinity to cynomolgus monkey MCHR1	Macaca fascicularis	1	ALA3856239	assay format	Scientific Literature
19.	ALA3858625	B	Binding affinity to rat MCHR1	Rattus norvegicus	2	ALA3856239	single protein format	Scientific Literature
20.	ALA3858632	A	Inhibition of CYP1A2 (unknown origin)	Homo sapiens	1	ALA3856239	single protein format	Scientific Literature