| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2149642 | B | Inhibition of PIM1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 2 hrs by electrophoretic mobility shift assay | 14 | ALA2146430 | single protein format | Scientific Literature | ||
| 2. | ALA2149643 | B | Inhibition of FLT3 at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 3. | ALA2149644 | B | Inhibition of PDGFRalpha at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 4. | ALA2149645 | B | Inhibition of SYK at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 5. | ALA2149646 | B | Inhibition of GSK3beta at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 6. | ALA2149647 | B | Inhibition of EGFR at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 7. | ALA2149648 | B | Inhibition of KDR at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 8. | ALA2149649 | B | Inhibition of Aurora A at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 9. | ALA2149650 | B | Inhibition of MLK1 at 22500 nM by ELISA | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 10. | ALA2149651 | B | Inhibition of MST1 at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 11. | ALA2149982 | B | Inhibition of PIM1 at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 12. | ALA2149983 | B | Inhibition of PIM2 at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 13. | ALA2149984 | B | Inhibition of PIM3 at 22500 nM by electrophoretic mobility shift assay | 1 | ALA2146430 | single protein format | Scientific Literature | ||
| 14. | ALA2149343 | A | Metabolic stability in human liver microsomes assessed as compound remaining at 1 uM after 1 hr | Homo sapiens | 4 | ALA2146430 | microsome format | Scientific Literature | |
| 15. | ALA2149344 | A | Metabolic stability in mouse liver microsomes assessed as compound remaining at 1 uM after 1 hr | Mus musculus | 4 | ALA2146430 | microsome format | Scientific Literature | |
| 16. | ALA5237807 | B | Inhibition of full length human PIM1 expressed in Escherichia coli BL21 (DE3) preincubated for 0.5 hrs followed by substrate addition and measured after 0.5 hrs using ARKRRRHPSGPPTA and ATP as substrate by Glo-kinase assay | Homo sapiens | 1 | ALA5236572 | assay format | Scientific Literature |
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