# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2166323 | Binding | Inhibition of trypsin at 25 uM assessed as Kinact/Ki ratio incubated for 15 mins by spectrofluorometry | 52 | ALA2163241 | assay format | Scientific Literature | ||
2. | ALA2166324 | Binding | Inhibition of chymotrypsin at 25 uM assessed as Kinact/Ki ratio incubated for 15 mins by spectrofluorometry | 52 | ALA2163241 | assay format | Scientific Literature | ||
3. | ALA2166325 | Binding | Inhibition of porcine pancreatic elastase at 25 uM assessed as Kinact/Ki ratio incubated for 15 mins by spectrofluorometry | Sus scrofa | 52 | ALA2163241 | protein format | Scientific Literature | |
4. | ALA2166326 | Binding | Inhibition of human leukocyte elastase at 25 uM assessed as Kinact/Ki ratio incubated for 15 mins by spectrofluorometry | Homo sapiens | 52 | ALA2163241 | single protein format | Scientific Literature | |
5. | ALA4256412 | Binding | Irreversible inhibition of human leukocyte elastase assessed as ratio of Kinact to Ki using MeO-Suc-Ala-Ala-Pro-Val-pNA as substrate by spectrophotometric method | Homo sapiens | 2 | ALA4251738 | single protein format | Scientific Literature | |
6. | ALA4256413 | Binding | Irreversible inhibition of human leukocyte elastase assessed as ratio of Kinact to Ki using MeO-Suc-Ala-Ala-Pro-Val-pNA as substrate incubated over 60 mins by spectrophotometric method | Homo sapiens | 4 | ALA4251738 | single protein format | Scientific Literature | |
7. | ALA4256414 | Binding | Inhibition of porcine pancreatic elastase assessed as ratio of Kinact to Ki using MeO-Suc-Ala-Ala-Pro-Val-pNA as substrate incubated over 60 mins by spectrophotometric method | Sus scrofa | 2 | ALA4251738 | protein format | Scientific Literature | |
8. | ALA4256416 | Binding | Inhibition of bovine factor 10a assessed as product formation at 1 uM using Boc-Ile-Glu-Gly-Arg-AMC as substrate incubated over 60 mins by fluorimetric method | Bos taurus | 3 | ALA4251738 | single protein format | Scientific Literature | |
9. | ALA4256417 | Binding | Inhibition of human thrombin assessed as product formation at 1 uM using Z-Gly-Gly-Arg-AMC as substrate incubated over 60 mins by fluorimetric method | Homo sapiens | 3 | ALA4251738 | single protein format | Scientific Literature | |
10. | ALA4256418 | Binding | Inhibition of bovine trypsin assessed as product formation at 1 uM using Suc-Ala-Ala-Pro-Arg-pNA as substrate incubated over 60 mins by spectrophotometric method | Bos taurus | 3 | ALA4251738 | assay format | Scientific Literature | |
11. | ALA4256419 | Binding | Inhibition of human cathepsin B assessed as product formation at 1 uM using Z-Arg-Arg-pNA as substrate incubated over 60 mins by spectrophotometric method | Homo sapiens | 3 | ALA4251738 | single protein format | Scientific Literature | |
12. | ALA4256420 | Binding | Inhibition of human cathepsin L assessed as product formation at 1 uM using Z-Phe-Arg-pNA as substrate incubated over 60 mins by spectrophotometric method | Homo sapiens | 3 | ALA4251738 | single protein format | Scientific Literature | |
13. | ALA4256422 | Binding | Inhibition of bovine chymotrypsin assessed as product formation at 1 uM using Suc-Ala-Ala-Pro-Phe-pNA as substrate incubated over 60 mins by spectrophotometric method | Bos taurus | 2 | ALA4251738 | assay format | Scientific Literature | |
14. | ALA4256426 | Binding | Irreversible inhibition of human leukocyte elastase at 20 nM using MeO-Suc-Ala-Ala-Pro-Val-pNA as substrate incubated for 30 mins followed by substrate addition | Homo sapiens | 1 | ALA4251738 | single protein format | Scientific Literature |