| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2167729 | B | Inhibition of [3H]R-(-)-14-induced receptor photolabeling at human FLAG-tagged alpha1 GABA A receptor expressed in HEK293S cells at 200 uM relative to untreated control | Homo sapiens | 1 | ALA2163302 | cell-based format | Scientific Literature | |
| 2. | ALA2167730 | B | Inhibition of [3H]R-(-)-14-induced receptor photolabeling at human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cells at 200 uM relative to untreated control | Homo sapiens | 1 | ALA2163302 | cell-based format | Scientific Literature | |
| 3. | ALA2168415 | B | Displacement of [3H]R-(-)-14 from human FLAG-tagged alpha1 GABA A receptor expressed in HEK293S cells | Homo sapiens | 3 | ALA2163302 | cell-based format | Scientific Literature | |
| 4. | ALA2168416 | B | Displacement of [3H]R-(-)-14 from human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cells | Homo sapiens | 3 | ALA2163302 | cell-based format | Scientific Literature | |
| 5. | ALA2168418 | B | Activation of human alpha1beta3gamma2L GABA A receptor expressed in HEK293 cells assessed as increase in [3H]muscimol binding by scintillation counting assay | Homo sapiens | 2 | ALA2163302 | cell-based format | Scientific Literature | |
| 6. | ALA2168419 | F | Agonist activity at human alpha1beta2gamma2L GABA A receptor expressed in Xenopus laevis oocytes assessed as increase in current response by two-electrode voltage clamp assay relative to GABA | Homo sapiens | 2 | ALA2163302 | cell-based format | Scientific Literature | |
| 7. | ALA2168420 | F | Agonist activity at human alpha1beta2gamma2L GABA A receptor expressed in Xenopus laevis oocytes assessed as increase in current response by two-electrode voltage clamp assay | Homo sapiens | 2 | ALA2163302 | cell-based format | Scientific Literature | |
| 8. | ALA2168421 | B | Activation of human alpha1beta2gamma2L GABA A receptor expressed in Xenopus laevis oocytes assessed as leftward shifting of GABA-induced current response at 8 uM by two-electrode voltage clamp assay relative to untreated control | Homo sapiens | 1 | ALA2163302 | cell-based format | Scientific Literature | |
| 9. | ALA2168422 | B | Activation of human alpha1beta2gamma2L GABA A receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced current response by two-electrode voltage clamp assay | Homo sapiens | 1 | ALA2163302 | cell-based format | Scientific Literature | |
| 10. | ALA2168644 | B | Activation of human alpha1beta2gamma2L GABA A receptor expressed in Xenopus laevis oocytes assessed as potentiation of 1000 uM GABA-induced current response at 8 uM by two-electrode voltage clamp assay relative to untreated control | Homo sapiens | 1 | ALA2163302 | cell-based format | Scientific Literature | |
| 11. | ALA2168647 | B | Activation of human alpha1beta2gamma2L GABA A receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced current response at 10 to 30 uM by two-electrode voltage clamp assay relative to untreated control | Homo sapiens | 1 | ALA2163302 | cell-based format | Scientific Literature | |
| 12. | ALA2168649 | F | Anesthetic activity in Xenopus laevis tadpoles assessed as loss of of righting reflexes | Xenopus laevis | 3 | ALA2163302 | organism-based format | Scientific Literature | |
| 13. | ALA2168652 | B | Activation of human alpha1beta2gamma2L GABA A receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced current response at 8 uM by two-electrode voltage clamp assay relative to untreated control | Homo sapiens | 1 | ALA2163302 | cell-based format | Scientific Literature |
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