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| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source |
| 1. | ALA2168707 | B | Selectivity ratio of IC50 for human recombinant CatB to IC50 for human recombinant CatK | Homo sapiens | 2 | | assay format | Scientific Literature |
| 2. | ALA2168708 | B | Inhibition of human recombinant CatK assessed as suppression of enzyme-mediated Z-Phe-Arg-AMC cleavage incubated for 1 hrs by QFRET assay | Homo sapiens | 38 | | single protein format | Scientific Literature |
| 3. | ALA2168709 | B | Inhibition of human recombinant CatL assessed as suppression of enzyme-mediated Z-Phe-Arg-AMC cleavage by QFRET assay | Homo sapiens | 33 | | single protein format | Scientific Literature |
| 4. | ALA2168710 | B | Inhibition of human recombinant CatS assessed as suppression of enzyme-mediated Z-Val-Val-Arg-AMC cleavage by QFRET assay | Homo sapiens | 36 | | single protein format | Scientific Literature |
| 5. | ALA2168711 | B | Inhibition of human recombinant CatB assessed as suppression of enzyme-mediated Z-Arg-Arg-AMC cleavage by QFRET assay | Homo sapiens | 34 | | single protein format | Scientific Literature |
| 6. | ALA2168712 | B | Inhibition of dog recombinant CatK assessed as suppression of enzyme-mediated Z-Phe-Arg-AMC cleavage by QFRET assay | Canis lupus familiaris | 1 | | single protein format | Scientific Literature |
| 7. | ALA2168713 | P | Lipophilicity, log D of the compound at pH 7.4 | | 32 | | small-molecule physicochemical format | Scientific Literature |
| 8. | ALA2168714 | A | Intrinsic clearance in dog hepatocytes assessed as metabolic turnover measured per 10'6 cells | Canis lupus familiaris | 3 | | cell-based format | Scientific Literature |
| 9. | ALA2168715 | A | Plasma clearance in Alderley Park Han Wistar rat at 2.0 mg/kg, po and 2.0 mg/kg, iv administered as single dose | Rattus norvegicus | 3 | | organism-based format | Scientific Literature |
| 10. | ALA2168716 | A | Plasma clearance in Beagle dog at 1.0 mg/kg, po and 1.0 mg/kg, iv administered as single dose | Canis lupus familiaris | 3 | | organism-based format | Scientific Literature |
| 11. | ALA2168717 | A | Volume of distribution at steady state in Alderley Park Han Wistar rat at 2.0 mg/kg, po and 2.0 mg/kg, iv administered as single dose | Rattus norvegicus | 3 | | organism-based format | Scientific Literature |
| 12. | ALA2168917 | A | Volume of distribution at steady state in Beagle dog at 1.0 mg/kg, po and 1.0 mg/kg, iv administered as single dose | Canis lupus familiaris | 3 | | organism-based format | Scientific Literature |
| 13. | ALA2168918 | A | Half life in Alderley Park Han Wistar rat at 2.0 mg/kg, iv administered as single dose | Rattus norvegicus | 3 | | organism-based format | Scientific Literature |
| 14. | ALA2168919 | A | Half life in Beagle dog at 1.0 mg/kg, iv administered as single dose | Canis lupus familiaris | 3 | | organism-based format | Scientific Literature |
| 15. | ALA2168920 | A | Oral bioavailability in Alderley Park Han Wistar rat at 2.0 mg/kg administered as single dose | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 16. | ALA2168921 | A | Oral bioavailability in Beagle dog at 2.0 mg/kg administered as single dose | Canis lupus familiaris | 3 | | organism-based format | Scientific Literature |
| 17. | ALA2168922 | F | In-vivo inhibition of CatK in orally dosed Alderley Park Beagle dog assessed as reduction in CTX-1 level at 0.1 to 2 mg/kg, po qd by ELISA | Canis lupus familiaris | 1 | | organism-based format | Scientific Literature |
| 18. | ALA2168923 | B | Inhibition at human ERG by ion works screening assay | Homo sapiens | 1 | | single protein format | Scientific Literature |
| 19. | ALA2168924 | A | Fraction unbound in human serum | Homo sapiens | 3 | | cell-free format | Scientific Literature |
| 20. | ALA2168925 | A | Intrinsic clearance in human hepatocytes assessed as metabolic turnover measured per 10'6 cells | Homo sapiens | 3 | | cell-based format | Scientific Literature |