| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2167991 | Binding | Inhibition of TACE using Mca-PLAQAV-Dpa-RSSSR-NH2 as substrate preincubated 15 mins measured every 30 sec for 30 mins | 7 | ALA2163235 | single protein format | Scientific Literature | ||
| 2. | ALA2167992 | Binding | Inhibition of human ADAMTS-5 expressed in CHO cells using WAAG-3R as substrate preincubated for 15 mins measured after 1 hr by FRET assay | Homo sapiens | 54 | ALA2163235 | cell-based format | Scientific Literature | |
| 3. | ALA2167993 | Binding | Inhibition of ADAMTS-4 using WAAG-3R as substrate preincubated for 15 mins measured after 1 hr | 7 | ALA2163235 | single protein format | Scientific Literature | ||
| 4. | ALA2167994 | Binding | Inhibition of MMP-13 using 5-FAM-TPGPLGL[Dap- (DNP)]ARRK(5-TAMRA)-amide as substrate after 45 mins | 7 | ALA2163235 | single protein format | Scientific Literature | ||
| 5. | ALA2167995 | Binding | Inhibition of ADAMTS-1 using FAM (5-carbosyfluorescein)-AE*LQGRPISIAK substrate after 2 hrs | 7 | ALA2163235 | single protein format | Scientific Literature | ||
| 6. | ALA2168191 | Binding | Selectivity ratio of IC50 for human ADAMTS-5 over IC50 for ADAMTS-1 | Homo sapiens | 6 | ALA2163235 | assay format | Scientific Literature | |
| 7. | ALA2168192 | Binding | Selectivity ratio of IC50 for human ADAMTS-5 over IC50 for MMP-13 | Homo sapiens | 6 | ALA2163235 | assay format | Scientific Literature | |
| 8. | ALA2168193 | Binding | Selectivity ratio of IC50 for human ADAMTS-5 over IC50 for TACE | Homo sapiens | 6 | ALA2163235 | assay format | Scientific Literature | |
| 9. | ALA2168194 | Binding | Selectivity ratio of IC50 for human ADAMTS-5 over IC50 for ADAMTS-4 | Homo sapiens | 6 | ALA2163235 | assay format | Scientific Literature |
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