# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2185152 | Binding | Inhibition of MAPK11 assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
2. | ALA2185153 | Binding | Inhibition of KIAA0551 assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
3. | ALA2185154 | Binding | Inhibition of STK36 assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
4. | ALA2185155 | Binding | Inhibition of SRC assessed as residual activity at 1000 nM | 1 | ALA2176950 | single protein format | Scientific Literature | ||
5. | ALA2185156 | Binding | Inhibition of RIPK2 assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
6. | ALA2185157 | Binding | Inhibition of MAPK14 assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
7. | ALA2185158 | Binding | Inhibition of GAK assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
8. | ALA2185159 | Binding | Inhibition of EGFR assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
9. | ALA2185160 | Binding | Inhibition of CSNK1E assessed as residual activity at 1000 nM | 2 | ALA2176950 | single protein format | Scientific Literature | ||
10. | ALA2185573 | Binding | Ratio of SB203580 IC50 to compound IC50 for inhibition of p38alpha MAPK | 16 | ALA2176950 | single protein format | Scientific Literature | ||
11. | ALA2185574 | Binding | Inhibition of p38alpha MAPK | 16 | ALA2176950 | single protein format | Scientific Literature | ||
12. | ALA4052478 | ADME | Inhibition of recombinant human GST-tagged wild type EGFR ( 668 to 1210 residues) cytoplasmic domain expressed in baculovirus expression system preincubated for 20 mins followed by addition of [33P]-ATP measured after 2 hrs by filter-binding method | Homo sapiens | 26 | ALA4049460 | assay format | Scientific Literature | |
13. | ALA4052479 | Binding | Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system preincubated for 20 mins followed by addition of [33P]-ATP measured after 2 hrs by filter-binding method | Homo sapiens | 26 | ALA4049460 | assay format | Scientific Literature | |
14. | ALA4052480 | Binding | Inhibition of recombinant human GST-tagged EGFR L858R/T790M double mutant cytoplasmic domain expressed in baculovirus expression system preincubated for 20 mins followed by addition of [33P]-ATP measured after 2 hrs by filter-binding method | Homo sapiens | 26 | ALA4049460 | assay format | Scientific Literature | |
15. | ALA5143770 | Binding | Inhibition of wild type EGFR (unknown origin) | Homo sapiens | 22 | ALA5143505 | single protein format | Scientific Literature |