| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA828923 | B | Inhibition constant against synaptosomal Mu opioid receptor | 5 | assay format | Scientific Literature | |||
| 2. | ALA829550 | B | Inhibition constant against synaptosomal Delta Opioid Receptor | 5 | assay format | Scientific Literature | |||
| 3. | ALA830764 | B | Selectivity for synaptosomal Delta than Mu Opioid Receptors | 3 | protein format | Scientific Literature | |||
| 4. | ALA834112 | F | Agonist activity against mu opioid receptor of guinea pig ileum | Cavia porcellus | 5 | tissue-based format | Scientific Literature | ||
| 5. | ALA833129 | F | Agonistic activity against delta opioid receptor of mouse vas deferens assay | Mus musculus | 5 | tissue-based format | Scientific Literature | ||
| 6. | ALA2188205 | F | Ratio of morphine to compound for antinociceptive activity in CD1 mouse at 1 umol/kg, sc | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 7. | ALA2188207 | F | Antinociceptive activity in sc dosed CD1 mouse assessed as thermal-stimulus induced tail flick latency after 6 to 7 hrs | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 8. | ALA2188212 | F | Antinociceptive activity in sc dosed CD1 mouse assessed as thermal-stimulus induced tail flick latency after 2 hrs relative to morphine | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 9. | ALA2188213 | F | Antinociceptive activity in sc dosed CD1 mouse assessed as thermal-stimulus induced tail flick latency after 2 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 10. | ALA2188214 | F | Antinociceptive activity in CD1 mouse assessed as AUC of thermal-stimulus induced tail flick latency assessed per min at 1 umol/kg, ip up to 120 mins | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 11. | ALA2188218 | F | Antinociceptive activity in CD1 mouse assessed as thermal-stimulus induced tail flick latency at 1 umol/kg, ip after 60 mins | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 12. | ALA2188639 | F | Antinociceptive activity in CD1 mouse assessed as thermal-stimulus induced tail flick latency at 1 umol/kg, ip up to 120 mins | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 13. | ALA2188640 | A | Metabolic stability in mouse plasma assessed as compound recovery after 2 hrs | Mus musculus | 6 | cell-free format | Scientific Literature | ||
| 14. | ALA2188641 | A | Metabolic stability in mouse brain assessed as compound recovery after 2 hrs | Mus musculus | 6 | tissue-based format | Scientific Literature | ||
| 15. | ALA2188642 | A | Biodistribution in ICR-CD1 mouse serum at 30000 cpm/uL, iv after 15 mins | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 16. | ALA2188643 | A | Biodistribution in ICR-CD1 mouse kidney at 30000 cpm/uL, iv | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 17. | ALA2188645 | A | Blood brain barrier transport in ICR-CD1 mouse brain assessed as parenchyma fraction at 30000 cpm/uL, iv | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 18. | ALA2188646 | A | Blood brain barrier transport in ICR-CD1 mouse brain assessed as brain efflux rate coefficient at 30000 cpm/uL, iv | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 19. | ALA2188647 | A | Blood brain barrier transport in ICR-CD1 mouse brain assessed as capillary fraction at 30000 cpm/uL, iv | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 20. | ALA2188648 | A | Apparent volume of distribution in ICR-CD1 mouse brain at 30000 cpm/uL, iv | Mus musculus | 6 | organism-based format | Scientific Literature |
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