| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2208544 | B | Inhibition of human GAT1 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 2. | ALA2208545 | B | Inhibition of human BGT1 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA2208546 | B | Inhibition of human GAT2 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA2208547 | B | Inhibition of human GAT3 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA2208548 | B | Inhibition of mouse GAT1 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA2208549 | B | Inhibition of mouse GAT2 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA2208550 | B | Inhibition of mouse GAT3 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA2208551 | B | Inhibition of mouse GAT4 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA2208552 | B | Inhibition of GAT1 in NMRI mouse astrocytes assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA2208553 | B | Inhibition of GAT2 in NMRI mouse astrocytes assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA2208554 | B | Inhibition of GAT3 in NMRI mouse astrocytes assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA2208555 | B | Inhibition of GAT4 in NMRI mouse astrocytes assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA2208556 | B | Inhibition of GAT1 in NMRI mouse cortical neurons assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 14. | ALA2208557 | B | Inhibition of GAT2 in NMRI mouse cortical neurons assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 15. | ALA2208558 | B | Inhibition of GAT3 in NMRI mouse cortical neurons assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 16. | ALA2208559 | B | Inhibition of GAT4 in NMRI mouse cortical neurons assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by liquid scintillation counting | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 17. | ALA2208560 | B | Displacement of [3H]GABA from GABAB receptor in Sprague-Dawley rat synaptic membrane at 100 uM after 60 mins by scintillation counting | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 18. | ALA2208561 | F | Agonist activity at human rho1 GABAc receptor expressed in xenopus laevis oocyte at 100 uM by electrophysiological method | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA2208562 | F | Antagonist activity at human rho1 GABAc receptor expressed in xenopus laevis oocyte assessed as inhibition of GABA-induced effect at 100 uM by electrophysiological method | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA2208563 | B | Inhibition of aspartate aminotransferase using L-aspartate as substrate at 6 mM incubated for 1 hr prior to substrate addition measured after 30 mins by spectrophotometric analysis | 1 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!