# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA684119 | B | Binding affinity determined by reduction in binding of 125 I-glucagon to the human glucagon receptor expressed on CHO cells in absence of Mg+2 | 47 | ALA1132135 | cell-based format | Scientific Literature | ||
2. | ALA684120 | B | Binding affinity towards glucagon receptor determined by reduction in binding of [125I]glucagon to the human glucagon receptor (GGR) expressed on CHO cells in presence of Mg+2 | 33 | ALA1132135 | cell-based format | Scientific Literature | ||
3. | ALA680807 | B | Binding affinity towards glucagon receptor determined by reduction in binding of [125I]glucagon to the murine glucagon receptor (GGR) expressed on CHO cells in absence of Mg+2 | 27 | ALA1132135 | cell-based format | Scientific Literature | ||
4. | ALA681685 | B | Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on CHO cells in presence of Mg+2 at 1 uM | 7 | ALA1132135 | cell-based format | Scientific Literature | ||
5. | ALA754535 | B | Inhibitory potency evaluated against rat p38 kinase | 53 | ALA1130598 | single protein format | Scientific Literature | ||
6. | ALA842195 | B | Inhibitory activity against p38-alpha kinase | 43 | ALA1132135 | single protein format | Scientific Literature | ||
7. | ALA845462 | B | Selectivity ratio between the binding value of human glucagon receptor (GGR) with Mg+2 and the value of p38 kinase | 25 | ALA1132135 | assay format | Scientific Literature | ||
8. | ALA884635 | F | Antagonist activity against glucagon receptor | Homo sapiens | 2 | ALA1140378 | assay format | Scientific Literature | |
9. | ALA881485 | B | Inhibitory activity against Mitogen-activated protein kinase 14, p38-alpha | Homo sapiens | 2 | ALA1140378 | single protein format | Scientific Literature | |
10. | ALA2437506 | B | Antagonist activity at human glucagon receptor | Homo sapiens | 35 | ALA2434841 | single protein format | Scientific Literature |