| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2320125 | B | Orthosteric antagonist activity at M5 muscarinic receptor in rat striatal slices assessed as inhibition of 100 uM oxotremorine-evoked [3H]DA release | Rattus norvegicus | 2 | assay format | Scientific Literature | ||
| 2. | ALA2320126 | B | Selectivity index, ratio of Ki for human M4 muscarinic receptor to Ki for human M5 muscarinic receptor | Homo sapiens | 9 | assay format | Scientific Literature | ||
| 3. | ALA2320127 | B | Selectivity index, ratio of Ki for human M3 muscarinic receptor to Ki for human M5 muscarinic receptor | Homo sapiens | 9 | assay format | Scientific Literature | ||
| 4. | ALA2320128 | B | Selectivity index, ratio of Ki for human M2 muscarinic receptor to Ki for human M5 muscarinic receptor | Homo sapiens | 9 | assay format | Scientific Literature | ||
| 5. | ALA2320129 | B | Displacement of [3H]NMS from human M4 muscarinic receptor expressed in CHO-K1 cells | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 6. | ALA2320130 | B | Displacement of [3H]NMS from human M3 muscarinic receptor expressed in CHO-K1 cells | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 7. | ALA2320131 | B | Displacement of [3H]NMS from human M2 muscarinic receptor expressed in CHO-K1 cells | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 8. | ALA2317404 | B | Orthosteric antagonist activity at human M5 muscarinic receptor expressed in CHO-K1 cells assessed as inhibition of [3H]NMS binding at saturation concentration relative to untreated control | Homo sapiens | 35 | cell-based format | Scientific Literature | ||
| 9. | ALA2317405 | B | Orthosteric antagonist activity at human M1 muscarinic receptor expressed in CHO-K1 cells assessed as inhibition of [3H]NMS binding at saturation concentration relative to untreated control | Homo sapiens | 35 | cell-based format | Scientific Literature | ||
| 10. | ALA2317406 | B | Selectivity index, ratio of Ki for human M1 muscarinic receptor to Ki for human M5 muscarinic receptor | Homo sapiens | 35 | assay format | Scientific Literature | ||
| 11. | ALA2317407 | B | Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cells | Homo sapiens | 60 | cell-based format | Scientific Literature | ||
| 12. | ALA2317408 | B | Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cells | Homo sapiens | 60 | cell-based format | Scientific Literature | ||
| 13. | ALA5164521 | B | Displacement of [3H]-NMS from human muscarinic M5 receptor expressed in CHO cells by radioligand binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 14. | ALA5164522 | B | Displacement of [3H]-NMS from human muscarinic M1 receptor expressed in CHO cells by radioligand binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA5164523 | B | Displacement of [3H]-NMS from human muscarinic M2 receptor expressed in CHO cells by radioligand binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA5164524 | B | Displacement of [3H]-NMS from human muscarinic M3 receptor expressed in CHO cells by radioligand binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA5164525 | B | Displacement of [3H]-NMS from human muscarinic M4 receptor expressed in CHO cells by radioligand binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature |
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