| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2317226 | B | Inhibition of CSNK1E (unknown origin) | Homo sapiens | 1 | ALA2311263 | single protein format | Scientific Literature | |
| 2. | ALA2317227 | B | Inhibition of p38beta MAP kinase (unknown origin) | Homo sapiens | 2 | ALA2311263 | single protein format | Scientific Literature | |
| 3. | ALA2317231 | B | Inhibition of p38alpha MAP kinase in whole blood (unknown origin) assessed as lipopolysaccharide-stimulated TNF-alpha release by ELISA | Homo sapiens | 46 | ALA2311263 | single protein format | Scientific Literature | |
| 4. | ALA2317232 | B | Inhibition of p38alpha MAP kinase (unknown origin) by ELISA | Homo sapiens | 48 | ALA2311263 | single protein format | Scientific Literature | |
| 5. | ALA4019401 | B | Inhibition of CSNK1E (unknown origin) at 1000 nM | Homo sapiens | 1 | ALA4017508 | single protein format | Scientific Literature | |
| 6. | ALA4019402 | B | Inhibition of P38 alpha MAPK (unknown origin) by ELISA | Homo sapiens | 70 | ALA4017508 | single protein format | Scientific Literature | |
| 7. | ALA4019403 | B | Binding affinity to wild type human biotin labelled p38 alpha (9 to 352 residues) expressed in sf21 insect cells SPR analysis | Homo sapiens | 12 | ALA4017508 | cell-based format | Scientific Literature | |
| 8. | ALA4019404 | B | Inhibition of P38 alpha MAPK in human whole blood assessed as reduction in TNF-alpha release after 10 mins by ELISA | Homo sapiens | 70 | ALA4017508 | single protein format | Scientific Literature | |
| 9. | ALA4019405 | B | Binding affinity to wild type biotin labelled human p38 alpha (9 to 352 residues) expressed in sf21 insect cells assessed as association rate constant by SPR analysis | Homo sapiens | 13 | ALA4017508 | cell-based format | Scientific Literature | |
| 10. | ALA4019406 | B | Binding affinity to wild type human biotin labelled p38 alpha (9 to 352 residues) expressed in sf21 insect cells assessed as dissociation rate constant by SPR analysis | Homo sapiens | 13 | ALA4017508 | cell-based format | Scientific Literature | |
| 11. | ALA4019407 | B | Binding affinity to wild type human biotin labelled p38 alpha (9 to 352 residues) expressed in sf21 insect cells assessed as residence time by SPR analysis | Homo sapiens | 12 | ALA4017508 | cell-based format | Scientific Literature | |
| 12. | ALA4019408 | B | Binding affinity to wild type human biotin labelled p38 alpha (9 to 352 residues) expressed in sf21 insect cells assessed as dissociation half life by SPR analysis | Homo sapiens | 12 | ALA4017508 | cell-based format | Scientific Literature | |
| 13. | ALA4019409 | A | Metabolic stability in rat liver microsomes after 180 mins in presence of NADPH by LC-MS analysis | Rattus norvegicus | 11 | ALA4017508 | assay format | Scientific Literature | |
| 14. | ALA4019410 | A | Drug metabolism in rat liver microsomes assessed as metabolite formation after 180 mins in presence of NADPH by LC-MS analysis | Rattus norvegicus | 11 | ALA4017508 | assay format | Scientific Literature | |
| 15. | ALA4618314 | B | Inhibition of recombinant human full-length N-terminal GST-tagged p38alpha MAPK expressed in baculovirus infected Sf9 insect cells using p38 peptide as substrate preincubated for 15 mins followed by substrate addition and measured after 60 mins by ADP-glo assay | Homo sapiens | 6 | ALA4616669 | cell-based format | Scientific Literature | |
| 16. | ALA4618315 | B | Inhibition of NanoBRET kinase tracer K4 binding to full-length human C-terminal NanoLuc-tagged p38alpha MAPK expressed in HEK293T cells incubated for 2 hrs by NanoBRET NanoGlo substrate based NanoBRET assay | Homo sapiens | 6 | ALA4616669 | cell-based format | Scientific Literature | |
| 17. | ALA4618316 | B | Inhibition of p38alpha MAPK in human whole blood assessed as reduction in LPS-induced TNFalpha production preincubated for 2.5 hrs followed by LPS stimulation by ELISA | Homo sapiens | 6 | ALA4616669 | tissue-based format | Scientific Literature | |
| 18. | ALA4618317 | B | Inhibition of p38alpha MAPK (unknown origin) assessed as target residence time using ATF2 as substrate preincubated for 1 hr followed by jump dilution in presence of substrate and measured every 3 mins for 4 hrs by TR-FRET assay | Homo sapiens | 7 | ALA4616669 | single protein format | Scientific Literature | |
| 19. | ALA4689845 | T | Multiplex assay against human fibroblast | Homo sapiens | 458 | ALA4689842 | cell-based format | EUbOPEN Chemogenomic Library | |
| 20. | ALA4689846 | T | Multiplex assay against HEK293T | Homo sapiens | 458 | ALA4689842 | cell-based format | EUbOPEN Chemogenomic Library |
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