| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2328716 | B | Inhibition of mPGES1 mediated PGE2 production in LPS-stimulated human whole blood by ELISA | Homo sapiens | 19 | single protein format | Scientific Literature | ||
| 2. | ALA2328717 | P | Solubility in phosphate buffer at pH 7.4 by nephelometric method | 19 | small-molecule physicochemical format | Scientific Literature | |||
| 3. | ALA2328718 | B | Inhibition of human mPGES1 by ELISA | Homo sapiens | 19 | single protein format | Scientific Literature | ||
| 4. | ALA2393802 | F | Antiinflammatory activity in Duncan Hartley guinea pig assessed as Inhibition of carrageenan-induced 6-keto-PGF1alpha production at 10 mg/kg, po | Cavia porcellus | 3 | organism-based format | Scientific Literature | ||
| 5. | ALA2393803 | F | Antiinflammatory activity in Duncan Hartley guinea pig assessed as Inhibition of carrageenan-induced PGE2 production at 10 mg/kg, po | Cavia porcellus | 4 | organism-based format | Scientific Literature | ||
| 6. | ALA2393804 | A | Plasma concentration in Duncan Hartley guinea pig at 10 mg/kg, po | Cavia porcellus | 4 | organism-based format | Scientific Literature | ||
| 7. | ALA2393805 | A | Oral bioavailability in Sprague-Dawley rat at 1 mg/kg | Rattus norvegicus | 5 | organism-based format | Scientific Literature | ||
| 8. | ALA2393806 | A | Mean residence time in Sprague-Dawley rat at 1 mg/kg, po | Rattus norvegicus | 7 | organism-based format | Scientific Literature | ||
| 9. | ALA2393807 | A | Half life in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 7 | organism-based format | Scientific Literature | ||
| 10. | ALA2393808 | A | Volume of distribution at steady state in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 7 | organism-based format | Scientific Literature | ||
| 11. | ALA2393809 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 16 | microsome format | Scientific Literature | ||
| 12. | ALA2393810 | A | Clearance in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 7 | organism-based format | Scientific Literature | ||
| 13. | ALA2393811 | B | Ratio of IC50 for mPGES-1 in healthy human whole blood to IC50 for mPGES-1 (unknown origin) | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 14. | ALA2393812 | B | Inhibition of mPGES-1-mediated PGE2 production in LPS-stimulated healthy human whole blood after 20 to 24 hrs by ELISA | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 15. | ALA2393934 | B | Inhibition of mPGES-1 (unknown origin) using PGH2 as substrate assessed as PGE2 synthesis by ELISA | Homo sapiens | 25 | single protein format | Scientific Literature |
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