| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2330004 | Binding | Binding affinity to Trypanosoma cruzi recombinant full length CYP51 by spectrophotometric analysis | Trypanosoma cruzi | 5 | ALA2321803 | assay format | Scientific Literature | |
| 2. | ALA2330005 | ADME | Permeability across human Caco2 cells | Homo sapiens | 1 | ALA2321803 | cell-based format | Scientific Literature | |
| 3. | ALA2330006 | Binding | Inhibition of human ERG at 10 uM relative to control | Homo sapiens | 1 | ALA2321803 | single protein format | Scientific Literature | |
| 4. | ALA2330007 | Binding | Inhibition of human ERG at 1 uM relative to control | Homo sapiens | 1 | ALA2321803 | single protein format | Scientific Literature | |
| 5. | ALA2330008 | ADME | Metabolic stability in human plasma after 1 to 4 hrs | Homo sapiens | 1 | ALA2321803 | cell-free format | Scientific Literature | |
| 6. | ALA2330009 | ADME | Plasma protein binding in human | Homo sapiens | 1 | ALA2321803 | cell-free format | Scientific Literature | |
| 7. | ALA2330010 | ADME | Metabolic stability in mouse plasma after 1 to 4 hrs | Mus musculus | 1 | ALA2321803 | cell-free format | Scientific Literature | |
| 8. | ALA2330011 | ADME | Plasma protein binding in mouse | Mus musculus | 1 | ALA2321803 | cell-free format | Scientific Literature | |
| 9. | ALA2330012 | ADME | Metabolic stability in human microsomes after 20 mins in presence of ketoconazole | Homo sapiens | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 10. | ALA2330013 | ADME | Metabolic stability in rat microsomes after 20 mins in presence of ketoconazole | Rattus norvegicus | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 11. | ALA2330014 | ADME | Metabolic stability in mouse microsomes after 20 mins in presence of ketoconazole | Mus musculus | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 12. | ALA2330015 | ADME | Metabolic stability in human microsomes after 20 mins in presence of quinidine | Homo sapiens | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 13. | ALA2330016 | ADME | Metabolic stability in rat microsomes after 20 mins in presence of quinidine | Rattus norvegicus | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 14. | ALA2330017 | ADME | Metabolic stability in mouse microsomes after 20 mins in presence of quinidine | Mus musculus | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 15. | ALA2330018 | ADME | Metabolic stability in human microsomes after 20 mins | Homo sapiens | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 16. | ALA2330019 | ADME | Metabolic stability in rat microsomes after 20 mins | Rattus norvegicus | 1 | ALA2321803 | microsome format | Scientific Literature | |
| 17. | ALA2330020 | Functional | Antitrypanosomal activity against Trypanosoma cruzi trypomastigote infected in mouse NIH/3T3 cells at 0.4 uM incubated for 3 days post infection by DAPI-staining based immunofluorescence assay | Trypanosoma cruzi | 1 | ALA2321803 | organism-based format | Scientific Literature | |
| 18. | ALA2330112 | Functional | Antitrypanosomal activity against Trypanosoma cruzi Y infected in monkey LLC-MK2 cells after 24 hrs by luciferase reporter gene assay | Trypanosoma cruzi | 1 | ALA2321803 | organism-based format | Scientific Literature | |
| 19. | ALA2330114 | Functional | Antitrypanosomal activity against Trypanosoma cruzi Tulahuen infected in monkey LLC-MK2 cells after 24 hrs by beta-galactosidase reporter gene assay | Trypanosoma cruzi | 1 | ALA2321803 | organism-based format | Scientific Literature | |
| 20. | ALA2330115 | ADME | Metabolic stability in mouse microsomes after 20 mins | Mus musculus | 1 | ALA2321803 | microsome format | Scientific Literature |
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