| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2327071 | A | Ratio of drug level in brain to plasma at steady state in rat at 1000 ng/g after 5 hrs | Rattus norvegicus | 6 | cell-free format | Scientific Literature | ||
| 2. | ALA2327072 | A | Ratio of drug level in brain to plasma in rat at 1 hr | Rattus norvegicus | 6 | cell-free format | Scientific Literature | ||
| 3. | ALA2327073 | A | Unbound fraction in rat brain at 1000 ng/g after 5 hrs by equilibrium dialysis method | Rattus norvegicus | 6 | tissue-based format | Scientific Literature | ||
| 4. | ALA2327074 | A | Unbound fraction in human plasma at 1000 ng/g after 5 hrs by equilibrium dialysis method | Homo sapiens | 2 | cell-free format | Scientific Literature | ||
| 5. | ALA2327075 | A | Unbound fraction in cynomolgus monkey plasma at 1000 ng/g after 5 hrs by equilibrium dialysis method | Macaca fascicularis | 2 | cell-free format | Scientific Literature | ||
| 6. | ALA2327076 | A | Unbound fraction in rhesus monkey plasma at 1000 ng/g after 5 hrs by equilibrium dialysis method | Macaca mulatta | 2 | cell-free format | Scientific Literature | ||
| 7. | ALA2327077 | A | Unbound fraction in rat plasma at 1000 ng/g after 5 hrs by equilibrium dialysis method | Rattus norvegicus | 6 | cell-free format | Scientific Literature | ||
| 8. | ALA2327078 | A | Efflux ratio of apparent permeability from basolateral to apical side over apical to basolateral side in human Caco2 cells at 20 uM | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 9. | ALA2327471 | A | Apparent permeability across apical to basolateral side in human Caco2 cells at 20 uM by LC-MS/MS analysis | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 10. | ALA2327473 | B | Selectivity ratio of Ki for rat alpha1D adrenoceptor to Ki for bovine alpha1A adrenoceptor | 1 | assay format | Scientific Literature | |||
| 11. | ALA2327474 | B | Selectivity ratio of Ki for hamster alpha1B adrenoceptor to Ki for bovine alpha1A adrenoceptor | 1 | assay format | Scientific Literature | |||
| 12. | ALA2327477 | B | Binding affinity to 5-HT2A receptor (unknown origin) by radioligand displacement assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA2327485 | B | Ratio of compound Ki to sertindole Ki for human dopamine D2 receptor | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 14. | ALA2327486 | B | Displacement of [3H]prazosine from rat alpha1D adrenoceptor expressed in CHO cells after 20 mins by scintillation counting analysis | Rattus norvegicus | 5 | cell-based format | Scientific Literature | ||
| 15. | ALA2327487 | B | Displacement of [3H]prazosine from hamster alpha1B adrenoceptor expressed in Rat1 cells after 20 mins by scintillation counting analysis | Mesocricetus auratus | 5 | cell-based format | Scientific Literature | ||
| 16. | ALA2327488 | B | Displacement of [3H]spiperone from human dopamine D2 receptor expressed in CHO cells after 30 mins by scintillation counting analysis | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
| 17. | ALA2327489 | B | Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysis | Bos taurus | 16 | cell-based format | Scientific Literature | ||
| 18. | ALA2327490 | B | Selectivity ratio of Ki for human dopamine D2 receptor to Ki for bovine alpha1A adrenoceptor | 16 | assay format | Scientific Literature |
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