# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA875513 | Functional | Tested for adenosine A2 receptor agonistic activity by determining coronary vasodilation | Cavia porcellus | 31 | ALA1126102 | assay format | Scientific Literature | |
2. | ALA640340 | Functional | Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum response | Cavia porcellus | 31 | ALA1126102 | assay format | Scientific Literature | |
3. | ALA640249 | Binding | Selectivity for A1 and A2 receptors was evaluated | Cavia porcellus | 31 | ALA1126102 | protein format | Scientific Literature | |
4. | ALA2327710 | Functional | Agonist activity at human recombinant adenosine A2A receptor expressed in CHO cells assessed as [3H]cAMP accumulation after 15 mins by liquid scintillation counting | Homo sapiens | 5 | ALA2321867 | cell-based format | Scientific Literature | |
5. | ALA2327711 | Binding | Selectivity ratio of Ki for human recombinant adenosine A1 receptor to Ki for adenosine A1 receptor in rat brain cortical membrane | 1 | ALA2321867 | cell membrane format | Scientific Literature | ||
6. | ALA2327712 | Binding | Selectivity ratio of Ki for human recombinant adenosine A2A receptor to Ki for adenosine A2A receptor in rat brain striatal membrane | 2 | ALA2321867 | cell membrane format | Scientific Literature | ||
7. | ALA2327844 | Binding | Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cells after 180 mins by liquid scintillation counting analysis | Homo sapiens | 18 | ALA2321867 | cell-based format | Scientific Literature | |
8. | ALA2328341 | Binding | Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells at 10 uM after 75 mins by liquid scintillation counting analysis | Homo sapiens | 18 | ALA2321867 | cell-based format | Scientific Literature | |
9. | ALA2328342 | Binding | Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells after 75 mins by liquid scintillation counting analysis | Homo sapiens | 18 | ALA2321867 | cell-based format | Scientific Literature | |
10. | ALA2328344 | Binding | Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in HEK cells | Homo sapiens | 4 | ALA2321867 | cell-based format | Scientific Literature | |
11. | ALA2328345 | Binding | Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membrane after 60 mins by liquid scintillation counting analysis | Rattus norvegicus | 20 | ALA2321867 | cell membrane format | Scientific Literature | |
12. | ALA2328348 | Binding | Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells 90 mins by liquid scintillation counting analysis | Homo sapiens | 2 | ALA2321867 | cell-based format | Scientific Literature | |
13. | ALA2328349 | Binding | Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by liquid scintillation counting analysis | Rattus norvegicus | 20 | ALA2321867 | cell membrane format | Scientific Literature |