| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2344111 | B | Inhibition of recombinant MAPKAPK2 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 2. | ALA2344113 | B | Inhibition of recombinant KDR (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 3. | ALA2344114 | B | Inhibition of recombinant MAPK14 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 4. | ALA2344115 | B | Inhibition of recombinant NEK1 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 5. | ALA2344116 | B | Inhibition of recombinant MEK1 (unknown origin) by cascade reaction assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 6. | ALA2344117 | B | Inhibition of recombinant ERK2 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 7. | ALA2344118 | B | Inhibition of recombinant RAF1 (unknown origin) by cascade reaction assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 8. | ALA2344119 | B | Inhibition of recombinant AMPK A1/B1/G1 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | protein complex format | Scientific Literature | ||
| 9. | ALA2344120 | B | Inhibition of recombinant RPS6K1 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 10. | ALA2344121 | B | Inhibition of recombinant AKT2 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 11. | ALA2344122 | B | Inhibition of recombinant IKBKB (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 12. | ALA2344124 | B | Inhibition of recombinant AKT1 (unknown origin) by FRET-based Z'-LYTE assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 13. | ALA3265869 | A | Drug metabolism in human liver S9 fraction assessed as (E)-1-methyl-3-(2-pyridinylmethyl)-5-(2-pyridinylmethylidene)-4-piperidone formation at 1 uM using 1% DMSO measured at 60 mins by LC/MS-MS analysis in presence of NADPH | Homo sapiens | 1 | subcellular format | Scientific Literature | ||
| 14. | ALA3265870 | A | Drug metabolism in human liver S9 fraction assessed as (E)-1-methyl-3,5-bis(2-pyridinylmethylidene)-4-hydroxypiperidine formation at 1 uM using 1% DMSO measured at 60 mins by LC/MS-MS analysis in presence of NADPH | Homo sapiens | 1 | subcellular format | Scientific Literature | ||
| 15. | ALA3265872 | F | Cytotoxicity against human TU212 cells assessed as cell viability at 5 to 10 uM after 48 hrs by neutral red dye uptake assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA3265874 | A | Half life in cynomolgus monkey liver S9 fraction at 1 uM using 1% DMSO | Macaca fascicularis | 1 | subcellular format | Scientific Literature | ||
| 17. | ALA3265875 | A | Half life in CD1 mouse liver S9 fraction at 1 uM using 1% DMSO | Mus musculus | 1 | subcellular format | Scientific Literature | ||
| 18. | ALA3265876 | A | Half life in human liver S9 fraction at 2 uM using 0.2% DMSO in presence of NADPH | Homo sapiens | 1 | subcellular format | Scientific Literature | ||
| 19. | ALA3265877 | A | Half life in human liver S9 fraction at 2 uM using 0.2% DMSO in absence of NADPH | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 20. | ALA3265879 | A | Metabolic stability in human liver S9 fraction assessed as remaining compound level at 2 uM using 0.2% DMSO measured after 1 hr by LC/MS-MS analysis in presence of NADPH | Homo sapiens | 1 | subcellular format | Scientific Literature |
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