| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2382553 | B | Reversible inhibition of human MAO-B using p-tyramine as substrate at IC80 incubated for 22 mins followed by substrate addition measured for 5 hrs by fluorescence assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 2. | ALA2382554 | B | Selectivity ratio of IC50 for MAO-B in mitochondria-enriched Sprague-Dawley rat liver fractions to IC50 for recombinant human MAO-B | 30 | mitochondrion format | Scientific Literature | |||
| 3. | ALA2382555 | B | Inhibition of recombinant human MAO-B expressed in baculovirus-infected insect cells using p-tyramine as substrate incubated for 30 mins prior to substrate addition measured for 45 mins by amplex red reagent-based microplate fluorescence reader analysis | Homo sapiens | 33 | cell-based format | Scientific Literature | ||
| 4. | ALA2382556 | B | Inhibition of MAO-B in mitochondria-enriched Sprague-Dawley rat liver fractions using p-tyramine as substrate incubated for 30 mins prior to substrate addition measured for 45 mins by amplex red reagent-based microplate fluorescence reader analysis | Rattus norvegicus | 33 | mitochondrion format | Scientific Literature | ||
| 5. | ALA2382684 | B | Selectivity ratio of Ki for human recombinant adenosine A1 receptor to Ki for human recombinant adenosine A2A receptor | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 6. | ALA2382685 | B | Selectivity ratio of Ki for human recombinant adenosine A3 receptor to Ki for human recombinant adenosine A2A receptor | Homo sapiens | 6 | assay format | Scientific Literature | ||
| 7. | ALA2382686 | B | Selectivity ratio of Ki for human recombinant adenosine A2B receptor to Ki for human recombinant adenosine A2A receptor | Homo sapiens | 6 | assay format | Scientific Literature | ||
| 8. | ALA2382687 | B | Selectivity ratio of Ki for adenosine A2A receptor in rat brain striatal membranes to Ki for human recombinant adenosine A2A receptor | 1 | cell membrane format | Scientific Literature | |||
| 9. | ALA2382690 | B | Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by liquid scintillation counting analysis | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 10. | ALA2382691 | B | Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells after 75 mins by liquid scintillation counting analysis | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 11. | ALA2382692 | B | Displacement of [3H]MSX2 from human recombinant adenosine A2A receptor expressed in CHO cells after 30 mins by liquid scintillation counting analysis | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 12. | ALA2382693 | B | Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells after 90 mins by liquid scintillation counting analysis | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 13. | ALA2382694 | B | Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membranes after 30 mins by liquid scintillation counting analysis | Rattus norvegicus | 30 | cell membrane format | Scientific Literature | ||
| 14. | ALA2382695 | B | Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranes after 90 mins by liquid scintillation counting analysis | Rattus norvegicus | 31 | cell membrane format | Scientific Literature |
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