| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2384809 | B | Selectivity ratio of IC50 for TNKS1 (unknown origin) to IC50 for TNKS2 PARP domain (947 to 1162) (unknown origin) | Homo sapiens | 1 | ALA2380224 | assay format | Scientific Literature | |
| 2. | ALA2384810 | B | Selectivity ratio of IC50 for PARP6 (unknown origin) to IC50 for TNKS2 PARP domain (947 to 1162) (unknown origin) | Homo sapiens | 1 | ALA2380224 | assay format | Scientific Literature | |
| 3. | ALA2384811 | B | Selectivity ratio of IC50 for PARP3 (unknown origin) to IC50 for TNKS2 PARP domain (947 to 1162) (unknown origin) | Homo sapiens | 1 | ALA2380224 | assay format | Scientific Literature | |
| 4. | ALA2384812 | B | Selectivity ratio of IC50 for PARP1 (unknown origin) to IC50 for TNKS2 PARP domain (947 to 1162) (unknown origin) | Homo sapiens | 1 | ALA2380224 | assay format | Scientific Literature | |
| 5. | ALA2382483 | B | Selectivity ratio of IC50 for PARP2 (unknown origin) to IC50 for TNKS2 PARP domain (947 to 1162) (unknown origin) | Homo sapiens | 1 | ALA2380224 | assay format | Scientific Literature | |
| 6. | ALA2382484 | B | Inhibition of PARP6 (unknown origin) | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 7. | ALA2382485 | B | Inhibition of PARP3 (unknown origin) | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 8. | ALA2382486 | B | Inhibition of TNKS1 (unknown origin) | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 9. | ALA2382487 | B | Inhibition of PARP1 (unknown origin) | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 10. | ALA2382488 | B | Inhibition of PARP2 (unknown origin) | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 11. | ALA2382489 | B | Inhibition of PARP7 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 12. | ALA2382490 | B | Inhibition of PARP11 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 13. | ALA2382491 | B | Inhibition of PARP6 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 14. | ALA2382492 | B | Inhibition of PARP2 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 15. | ALA2382493 | B | Inhibition of PARP3 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 16. | ALA2382494 | B | Inhibition of PARP1 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 17. | ALA2382496 | B | Inhibition of auto-PARsylation of GST-tagged TNKS2 PARP domain (947 to 1162) (unknown origin) expressed in Escherichia coli BL21(DE3) after 2 hrs by LC/MS analysis | Homo sapiens | 14 | ALA2380224 | assay format | Scientific Literature | |
| 18. | ALA2382498 | B | Binding affinity to TNKS2 PARP domain (947 to 1162) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as thermal stabilization at 125 uM by differential scanning flourimetric analysis | Homo sapiens | 11 | ALA2380224 | assay format | Scientific Literature | |
| 19. | ALA2382500 | B | Binding affinity to 6His-tagged TNKS2 PARP domain (947 to 1162) (unknown origin) expressed in Escherichia coli BL21(DE3) by surface plasmon resonance analysis | Homo sapiens | 6 | ALA2380224 | assay format | Scientific Literature |
The page will load shortly, Thanks for your patience!