| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2383556 | F | Inverse agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as increase in forskolin-stimulated cAMP production by scintillation counting analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 2. | ALA2383558 | F | Inverse agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as increase in forskolin-stimulated cAMP production at 10 uM by scintillation counting analysis relative to WIN55212-2 | Homo sapiens | 40 | cell-based format | Scientific Literature | ||
| 3. | ALA2383559 | F | Inverse agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as increase in forskolin-stimulated cAMP production at 1 uM by scintillation counting analysis relative to WIN55212-2 | Homo sapiens | 40 | cell-based format | Scientific Literature | ||
| 4. | ALA2383560 | B | Selectivity index, ratio of Ki for human CB1 receptor to Ki for human CB2 receptor | Homo sapiens | 41 | assay format | Scientific Literature | ||
| 5. | ALA2383561 | B | Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membrane after 60 mins by scintillation counting analysis | Homo sapiens | 41 | cell-based format | Scientific Literature | ||
| 6. | ALA2383562 | B | Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cell membrane after 90 mins by scintillation counting analysis | Homo sapiens | 41 | cell-based format | Scientific Literature | ||
| 7. | ALA2383563 | B | Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cell membrane at > 10 uM after 90 mins by scintillation counting analysis | Homo sapiens | 27 | cell-based format | Scientific Literature | ||
| 8. | ALA2383564 | B | Displacement of [3H]CP-55940 from Sprague-Dawley rat brain CB1 receptor at > 10 uM after 90 mins by scintillation counting analysis | Rattus norvegicus | 27 | assay format | Scientific Literature | ||
| 9. | ALA2383565 | B | Displacement of [3H]CP-55940 from Sprague-Dawley rat brain CB1 receptor after 90 mins by scintillation counting analysis | Rattus norvegicus | 41 | assay format | Scientific Literature | ||
| 10. | ALA2383566 | B | Displacement of [3H]CP-55940 from Sprague-Dawley rat spleen CB2 receptor after 60 mins by scintillation counting analysis | Rattus norvegicus | 41 | single protein format | Scientific Literature |
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