| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2390099 | B | Selectivity ratio of Kinact for human liver cathepsin B to Kinact for human cathepsin D | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 2. | ALA2390100 | B | Selectivity ratio of Kinact for human liver cathepsin B to Kinact for human cathepsin S | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 3. | ALA2390101 | B | Selectivity ratio of Kinact for human liver cathepsin B to Kinact for human cathepsin F | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA2388369 | B | Inhibition of cathepsin in human MDA-MB-231 cells assessed as decrease in cell migratory behavior after 6 hrs by microscopic analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA2388370 | B | Inhibition of cathepsin S in human MDA-MB-231 cells assessed as increase in E-cadherin levels at 1 to 5 uM after 30 mins by Western blotting analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA2388371 | B | Inhibition of cathepsin B in human MDA-MB-231 cells assessed as increase in E-cadherin levels at 1 to 5 uM after 30 mins by Western blotting analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA2388372 | B | Inhibition of cathepsin in human MDA-MB-231 cells assessed as change in cellular morphology at 20 uM by microscopic analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA2388373 | B | Inhibition of cathepsin S in human MDA-MB-231 cells assessed as increase in E-cadherin levels after 20 mins by immunofluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA2388374 | B | Inhibition of cathepsin B in human MDA-MB-231 cells assessed as increase in E-cadherin levels after 20 mins by immunofluorescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA2388375 | B | Inhibition of cathepsin B in human MDA-MB-231 cells using Z-RR-AMC as substrate preincubated for 20 mins prior to substrate addition measured after 10 mins by confocal microscopic analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA2388549 | P | Half life of the compound at 2.5 mM at pH 7.4 by NMR spectrophotometric analysis | 1 | small-molecule physicochemical format | Scientific Literature | |||
| 12. | ALA2388550 | B | Inhibition of cathepsin B in human MDA-MB-231 cells using Z-RR-AMC as substrate at 20 uM preincubated for 20 mins prior to substrate addition measured after 10 mins by confocal microscopic analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA2388551 | B | Inhibition of human PTP1B | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA2388552 | B | Inhibition of trypsin (unknown origin) using N-alpha-benzoyl-DL-arginine-p-nitroanilide as substrate | Homo sapiens | 1 | protein format | Scientific Literature | ||
| 15. | ALA2388553 | B | Inhibition of human cathepsin G using Suc-AAPF-pNA as substrate | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA2388554 | B | Inhibition of human cathepsin D using Mca-Gly-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Lys(Dnp)-D-Arg-NH2 as substrate | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA2388555 | B | Inhibition of human cathepsin S using Z-VVR-AMC as substrate | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA2388556 | B | Inhibition of human cathepsin F using Z-FR-AMC as substrate | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA2388557 | B | Inhibition of human liver cathepsin B using Z-RR-para-nitroanilide as substrate | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA2388558 | B | Inhibition of human liver cathepsin B in presence of azide ion | Homo sapiens | 1 | assay format | Scientific Literature |
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