# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2404651 | B | Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from mouse adenosine A3 receptor expressed in HEK293 cell membranes after 60 mins by liquid scintillation counting analysis | Mus musculus | 10 | ALA2401698 | cell-based format | Scientific Literature | |
2. | ALA2404652 | B | Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5'-N-ethylcarboxamidoadenosine from mouse adenosine A2A receptor expressed in HEK293 cell membranes at 10 uM after 60 mins by liquid scintillation counting analysis relative to control | Mus musculus | 12 | ALA2401698 | cell-based format | Scientific Literature | |
3. | ALA2404653 | B | Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from mouse adenosine A1 receptor expressed in HEK293 cell membranes at 10 uM after 60 mins by liquid scintillation counting analysis relative to control | Mus musculus | 9 | ALA2401698 | cell-based format | Scientific Literature | |
4. | ALA2404655 | B | Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from human adenosine A3 receptor expressed in CHO cell membranes after 60 mins by liquid scintillation counting analysis | Homo sapiens | 5 | ALA2401698 | cell-based format | Scientific Literature | |
5. | ALA2404656 | B | Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5'-N-ethylcarboxamidoadenosine from human adenosine A2A receptor expressed in HEK293 cell membranes at 10 uM after 60 mins by liquid scintillation counting analysis relative to control | Homo sapiens | 5 | ALA2401698 | cell-based format | Scientific Literature | |
6. | ALA2404657 | B | Displacement of [3H]N6-R-phenylisopropyladenosine from human adenosine A1 receptor expressed in CHO cell membranes at 10 uM after 60 mins by liquid scintillation counting analysis relative to control | Homo sapiens | 4 | ALA2401698 | cell-based format | Scientific Literature | |
7. | ALA2403961 | F | Agonist activity at mouse adenosine A3 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP production preincubated for 30 mins prior to forskolin-treatment measured after 15 mins by ELISA relative to control | Mus musculus | 5 | ALA2401698 | cell-based format | Scientific Literature | |
8. | ALA2403962 | F | Agonist activity at mouse adenosine A3 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP production preincubated for 30 mins prior to forskolin-treatment measured after 15 mins by ELISA | Mus musculus | 4 | ALA2401698 | cell-based format | Scientific Literature | |
9. | ALA2403963 | F | Activity at mouse adenosine A3 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP production preincubated for 30 mins prior to forskolin-treatment measured after 15 mins by ELISA relative to 2-chloro-N6-(3-iodobenzyl)adenosine-5'-N-methyluronamide | Mus musculus | 12 | ALA2401698 | cell-based format | Scientific Literature | |
10. | ALA2403964 | F | Activity at human adenosine A3 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP production at 10 uM preincubated for 30 mins prior to forskolin-treatment measured after 15 mins by ELISA relative to 5'-N-ethylcarboxamidoadenosine | Homo sapiens | 5 | ALA2401698 | cell-based format | Scientific Literature | |
11. | ALA5155951 | B | Binding affinity to human adenosine A1A receptor expressed in human HEK293 cell membrane at 10 uM by radioligand inhibition assay | Homo sapiens | 28 | ALA5154659 | cell membrane format | Scientific Literature | |
12. | ALA5155952 | B | Binding affinity to mouse adenosine A1A receptor expressed in human HEK293 cell membrane by radioligand inhibition assay | Mus musculus | 9 | ALA5154659 | cell membrane format | Scientific Literature | |
13. | ALA5155953 | B | Binding affinity to human adenosine A2A receptor expressed in human HEK293 cell membrane at 10 uM by radioligand inhibition assay | Homo sapiens | 24 | ALA5154659 | cell membrane format | Scientific Literature | |
14. | ALA5155954 | B | Binding affinity to mouse adenosine A2A receptor expressed in human HEK293 cell membrane by radioligand inhibition assay | Mus musculus | 1 | ALA5154659 | cell membrane format | Scientific Literature | |
15. | ALA5155957 | B | Displacement of [125I] N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from human A3A receptor stably expressed in HEK293 cell membrane by radioligand inhibition assay | Homo sapiens | 31 | ALA5154659 | cell membrane format | Scientific Literature | |
16. | ALA5155979 | B | Displacement of [125I] N6-4-amino-3-iodobenzyl adenosine 5-N-methyluronamide from mouse A3A receptor stably expressed in HEK293 cell membrane by radioligand inhibition assay | Mus musculus | 25 | ALA5154659 | cell membrane format | Scientific Literature |